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- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
57186-25-1
- 规格:
10 mM * 1 mL/1 mg/5 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥4950.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥2045.0 |
| 规格: | 5 mg | 产品价格: | ¥4500.0 |
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Paxilline
CAS No. : 57186-25-1
MCE 国际站:Paxilline
产品活性:Paxilline 是一种来自 Penicillium paxilli 的吲哚生物碱霉菌毒素,通过封闭通道的阻断机制有效地抑制 BK 通道。 Paxilline 也能抑制肌质网 Ca2+ 刺激的 ATP 酶 (SERCA),对不同亚型的 SERCA 作用的 IC50 值为介于 5 μM-50 μM 之间。 Paxilline 具有显着的抗惊厥活性。
研究领域:Membrane Transporter/Ion Channel | Neuronal Signaling
作用靶点:Potassium Channel | Calcium Channel
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