- ￥590 - 5213
- MedChemExpress(MCE)
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- 2025年12月05日
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- 技术资料
- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名：
CVT-510
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
204512-90-3
- 规格：
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg
| 规格： | 10 mM * 1 mL | 产品价格： | ￥1104.0 |
|---|---|---|---|
| 规格： | 1 mg | 产品价格： | ￥590.0 |
| 规格： | 5 mg | 产品价格： | ￥1488.0 |
| 规格： | 10 mg | 产品价格： | ￥2225.0 |
| 规格： | 25 mg | 产品价格： | ￥3725.0 |
| 规格： | 50 mg | 产品价格： | ￥5213.0 |
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Tecadenoson
CAS No. : 204512-90-3
MCE 国际站：Tecadenoson
产品活性：Tecadenoson (CVT-510) 是选择性的腺苷受体 (A1 adenosine receptor) 激动剂。
研究领域：GPCR/G Protein
作用靶点：Adenosine Receptor
In Vitro: In the atrial-paced isolated heart, Tecadenoson is approximately 5 fold more potent to prolong the stimulus-to-His bundle (S-H interval), a measure of slowing AV nodal conduction (EC50=41 nM) than to increase coronary conductance (EC50=200 nM). At concentrations of Tecadenoson (40 nM) and diltiazem (1 μM) that causes equal prolongation of S-H interval (∼10 ms), diltiazem, but not Tecadenoson, significantly reduces left ventricular developed pressure (LVP) and markedly increases coronary conductance. Tecadenoson shortens atrial (EC50=73 nM) but not the ventricular monophasic action potentials (MAP).
In Vivo: In atrial-paced anaesthetized guinea-pigs, intravenous infusions of Tecadenoson and diltiazem causes nearly equal prolongations of P-R interval. Tecadenoson (2, 5, 20 μg/kg i.p.) causes a rapid and sustained dose-dependent decrease in NEFA at doses that do not cause bradycardia. Tecadenoson given at 50 μg/kg causes a significant bradycardia (50% decrease in heart rate at 25 min.
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