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- 详细信息
- 文献和实验
- 技术资料
- 库存:
170
- 英文名:
Scopolamine hydrobromide
- CAS号:
114-49-8
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|100mg|500mg
特别提示:包括muscarinic拮抗剂在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:muscarinic拮抗剂
英文名称:Scopolamine hydrobromide
产品货号:M05803
产品规格:1mL(10mM)|100mg|500mg
Scopolamine hydrobromide是高亲和力的(nM级别)毒蕈碱(muscarinic)拮抗剂。Scopolamine可逆抑制5-HT3受体反应,IC50为2.09μM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:114-49-8
别名:(-)-Scopolamine hydrobromide;Hyoscine hydrobromide;Scopine hydrobromide
纯度:98.0%
分子式:C₁₇H₂₂BrNO₄
分子量:384.26
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
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文献和实验Muscarinic Cholinergic Receptors
receptor population is divided between nicotinic and muscarinic subclasses, the CNS-associated cholinergic receptor appears to be predominantly of the muscarinic type, although there is evidence that the spinal cord contains substantial amounts of nicotinic
The vast majority of receptors are membrane proteins, so solubilization is an essential prerequisite for purification of these receptors. If the receptor can be solubilized without destroying its characteristic ability to bind specific
佚名 纳洛酮(naloxone)化学结构与吗啡极相似,主要区别为叔氮上以烯丙基取代甲基,6位羟基变为酮基(见表18-1)。纳洛酮对4型阿片受体都有拮抗作用(见表18-2)。它本身并无明显药理效应及毒性,给人注射12mg后,不产生任何症状;注射24mg只产生轻微困倦。但对吗啡中毒者,小剂量(0.4~0.8mg)肌内或静脉注射能迅速翻转吗啡的作用,1~
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