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- 询价记录
- 文献和实验
- 技术资料
- 保存条件:
4°C, sealed storage, away from moisture
- 英文名:
VUF 8325 dihydrobromide; SKF 91105 dihydrobromide
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
32385-58-3
- 规格:
1 mg/5 mg
| 规格: | 1 mg | 产品价格: | ¥460.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥1100.0 |
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Imetit dihydrobromide
CAS No. : 32385-58-3
MCE 国际站:Imetit dihydrobromide
产品活性:Imetit dihydrobromide (VUF 8325 dihydrobromide) 是组胺 H3 和 H4 受体的高亲和力的强激动剂,Ki 值分别为 0.3 和 2.7 nM。Imetit dihydrobromide 模拟组胺对嗜酸性粒细胞形状改变的作用 (EC50=25 nM)。
研究领域:GPCR/G Protein | Neuronal Signaling | Immunology/Inflammation
作用靶点:Histamine Receptor
In Vivo: Imetit dihydrobromide (2.5-10 mg/kg; i.p.) reduces the licking response induced by Apomorphine.
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文献和实验Characterization of Histaminergic Receptors
4 Agonists Histamine 6500 33,000 7.0 8.1 d Sigma Imetit 30,000 39,000 0.40 2.7 d RBI Immepip 22,000 >100,000 2.8 9.0 d Tocris Cookson
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