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- 详细信息
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
EU-5346
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
315698-17-0
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥1005.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥380.0 |
| 规格: | 5 mg | 产品价格: | ¥1100.0 |
| 规格: | 10 mg | 产品价格: | ¥1750.0 |
| 规格: | 25 mg | 产品价格: | ¥3038.0 |
| 规格: | 50 mg | 产品价格: | ¥4530.0 |
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ML311
CAS No. : 315698-17-0
MCE 国际站:ML311
产品活性:ML311 是 Mcl-1/Bim 蛋白之间相互作用的有效选择性抑制剂。
研究领域:Apoptosis
作用靶点:Bcl-2 Family
In Vitro: ML311 potently halts viability of several types of Mcl-1 primed cells, including MCL-1-1780 (EC50=0.31 μM), DHL-6 (EC50=3.3 μM), and NCI-H929 (EC50=1.6 μM), with generally high maximal effect (>80%). ML311 also displays activity in a leukemia-derived cell line particularly reliant upon Bcl-2 function (Bcl2-1863, EC50=1.1 μM). ML311 has strong growth inhibitory effects in many cell lines, with GI50<900 nM for nine cell types (RPMI-8226, SR, NCI-H322M, NCI-H60, HCC-2998, KM12, SF-295, U251, PC-3 cell lines), and <2 μM for 14 additional types.
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