- 询价
- MedChemExpress(MCE)
- 美国
- HY-U00353
- 2025年12月05日
企业认证
相关产品推荐更多 >
万千商家帮你免费找货
0 人在求购买到急需产品
- 详细信息
- 文献和实验
- 技术资料
- 保存条件：
Please store the product under the recommended conditions in the Certificate of Analysis.
- 库存：
货期：询盘
- 供应商：
MedChemExpress LLC
- CAS号：
391610-37-0
- 规格：
询盘
MCE 的所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务。
MCHR1 antagonist 1
CAS No. : 391610-37-0
MCE 国际站：MCHR1 antagonist 1
产品活性：MCHR1 antagonist 1 是一种选择性的黑色素浓集激素 1 型受体 (melanin concentrating hormone-1 receptor) 拮抗剂，对人 MCH1 受体的 Kb 和 Ki 值分别为 1 nM 和 4 nM，在降低体重方面可能起作用。
研究领域：GPCR/G Protein | Neuronal Signaling
作用靶点：MCHR1 (GPR24)
In Vitro: MCHR1 antagonist 1 shows potent activities against melanin concentrating hormone-1 receptor, but less potent against human MCH1, NPY1, NPY5, GALR1, GALR2, GALR3, and rat 5HT2C receptors, with Kis of >50000 nM.
相关产品：SNAP 94847 hydrochloride | Melanin Concentrating Hormone, salmon TFA | MCH(human, mouse, rat) TFA | AZD1979 | [Ala17]-MCH | ALB-127158(a) | Ethyl linolenate | GW-803430 | MCH-1 antagonist 1 | MCHR1 antagonist 2 | TC-MCH 7c | (Phe13,Tyr19)-MCH (human, mouse, rat) | Ac-hMCH(6-16)-NH2 | AMG-076 | ATC0175 | BMS-814580 | hMCH-1R antagonist 1 | MCHR1 antagonist 3 | Neuropeptide EI, rat | BMS-819881 | NGD-4715 | SB-568849
热门产品线：重组蛋白 | 化合物库 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物
Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Dye Reagents | PROTAC | Isotope-Labeled Compounds
风险提示：丁香通仅作为第三方平台，为商家信息发布提供平台空间。用户咨询产品时请注意保护个人信息及财产安全，合理判断，谨慎选购商品，商家和用户对交易行为负责。对于医疗器械类产品，请先查证核实企业经营资质和医疗器械产品注册证情况。
文献和实验Characterization of Histaminergic Receptors
(see De Backer et al., ) with human H 1 receptors using Lipofectamine 2000 (Life Technologies), grown to confluence Cell dissociation buffer (Life Technologies), prewarmed to 37°C Dulbecco's
[3H](+)MK801 Radioligand Binding Assay at the N‐Methyl‐D‐Aspartate Receptor
for agonist and antagonist compounds. (A ) These curves show the anticipated profile of a glycine site agonist added alone (open symbols) or in the presence (filled symbols) of the glycine site antagonist, 5,7‐dichlorokynurenate (5 µM). Data are modeled based
Characterization of Neurotensin Receptors
either radiolabeled neurotensin or SR 48692 (a nonpeptide neurotensin antagonist) as radioligands are described. These procedures may be used to screen selective ligands at neurotensin receptor subtypes. Keywords: neurotensin; SR 48692
技术资料暂无技术资料 索取技术资料
