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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1218816-71-7
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥3068.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥1400.0 |
| 规格: | 5 mg | 产品价格: | ¥3500.0 |
| 规格: | 10 mg | 产品价格: | ¥6000.0 |
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SK1-IN-1
CAS No. : 1218816-71-7
MCE 国际站:SK1-IN-1
产品活性:SK1-IN-1是一种有效的鞘氨醇激酶1 (SPHK1) 抑制剂,IC50 值为58 nM。
作用靶点:SphK
In Vivo: SK1-IN-1 demonstrates significant improvement in the intrinsic clearance, particularly against human liver microsomes. SK1-IN-1 is selected for rat PK studies and demonstrates modest in oral bioavailability with acceptable half-lives in blood circulation.
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文献和实验tkwggxOgYxdvEj687uNt8dWwWVYV2b9dxboxU7Fq4EyUvr4G9XJG91xREJIPdrhkmwVKsiD4/XSDp68KjDu1R+Ni2pIRqoJmwcMwgQxBgIWPDLGNvAgmkFEIqCJf7Z7oU6g4+pq3RmGhUTDoipkLb+JCH1vseeSNeg2yp8pis7RYj3MWtSCZocj84Lx/KNpMm4KJparjSP9CkkYkVSbGgzKBdEggFQ9M0yEtnjITYAIpTEADRbpMwcyJbUMFj7+jaeiZIDcC4P71
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