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- 详细信息
- 文献和实验
- 技术资料
- 库存:
69
- 英文名:
Narlaprevir
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|10mg|50mg|100mg
特别提示:包括NS3蛋白酶抑制剂(Narlaprevir)在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:NS3蛋白酶抑制剂(Narlaprevir)
英文名称:Narlaprevir
CAS#:865466-24-6
产品货号:NS3蛋白酶抑制剂(Narlaprevir)
产品规格:1mL(10mM)|10mg|50mg|100mg
Narlaprevir是NS3蛋白酶抑制剂,Ki为6nM,EC90为40nM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:865466-24-6
别名:SCH 900518
分子式:C₃₆H₆₁N₅O₇S
分子量:707.96
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
除了NS3蛋白酶抑制剂(Narlaprevir),SCH 900518,我公司还供应以下相关产品:
| 货号 | 名称 | 规格 |
| KFS297 | PD 98,059(MAPKK抑制剂) | 2mg |
| M00414 | 鞘氨醇激酶2抑制剂(SK2抑制剂)(ABC294640) | 1mL(10mM)|5mg|10mg|50mg|100mg |
| M00429 | Akt广谱抑制剂(Afuresertib) | 1mL(10mM)|2mg|5mg|10mg|50mg|100mg |
| M00558 | DT-diaphorase抑制剂(DMXAA) | 1mL(10mM)|5mg|10mg|50mg|100mg |
| M00919 | 泛Ras抑制剂(泛RAS-IN-1) | 1mL(10mM)|1mg|5mg|10mg|25mg|50mg|100mg |
| M00990 | GSK-3β抑制剂(CP21R7) | 1mL(10mM)|1mg|5mg|10mg |
| M01189 | GSK-3β抑制剂(TDZD-8) | 1mL(10mM)|10mg|50mg|100mg |
| M01205 | ALDH1A1抑制剂(NCT-501) | 1mL(10mM)|5mg|10mg|50mg|100mg |
| M01454 | CDK抑制剂(RGB-286638 free base) | 1mL(10mM)|2mg|5mg|10mg|50mg|100mg |
| M01539 | TRK家族受体抑制剂(LOXO-101 sulfate) | 1mL(10mM)|5mg|10mg|50mg|100mg |
| M01763 | GDH1抑制剂(R162) | 1mL(10mM)|5mg|10mg|25mg|50mg|100mg |
| M01971 | IDO抑制剂(IDO-IN-8) | 1mL(10mM)|1mg|5mg|10mg |
| M02201 | c-Met抑制剂(AMG-208) | 5mg|10mg|50mg|100mg |
| M03517 | NRTI和HIV-1抑制剂(Emtricitabine) | 1mL(10mM)|50mg|100mg|200mg|500mg |
| M04227 | 真菌抑制剂(Ravuconazole) | 1mL(10mM)|1mg|5mg|10mg|25mg|50mg |
| M04451 | 12-LOX抑制剂(ML355) | 1mL(10mM)|2mg|5mg|10mg|50mg|100mg |
| M05272 | DGAT1抑制剂(LCQ-908) | 1mL(10mM)|5mg|10mg|50mg |
| M05386 | GPR119激动剂(APD597) | 1mL(10mM)|5mg|10mg|50mg|100mg |
| M05739 | sodium channel抑制剂(Tetrodotoxin) | 1mg |
| M06222 | 碳酸*(代"酐")酶抑制剂(Dichlorphenamide) | 1mL(10mM)|10mg|50mg|100mg |
| M08142 | 乙酰辅酶A羧化酶抑制剂 | 1mL(10mM)|1mg|5mg |
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文献和实验Expression and Characterization of HCV NS3 Protease
The overexpression of a gene in a heterologous system is often the prelude to or the prerequisite of the elucidation and characterization of a given protein, in particular where the protein is difficult to obtain in sufficient quantity
Expression and Characterization of the HCV NS3 Helicase Domain
The hepatitis C virus (HCV) NS3 protein has two distinct biochemical domains. The N-terminal 20 kDa has serine protease activity (see Chapter 31 ) and the C-terminal 50 kDa has both nucleoside triphosphatase (NTPase) and helicase activities
蛋白 酶 已知对应的抑制剂 蛋白 酶 已知对应的抑制
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