Maropitant马罗皮坦,147116-67-4

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Maropitant

CAS No. : 147116-67-4

MCE 国际站：Maropitant

产品活性：Maropitant 是一种选择性的具有口服活性的神经激肽 (NK1 ) 受体拮抗剂。Maropitant 通过阻止催吐中心与化学感受器触发区 (CRTZ) 中 P 物质的结合而起作用。Maropitant 在预防呕吐方面非常有效。

研究领域：GPCR/G Protein  |  Neuronal Signaling

作用靶点：Neurokinin Receptor

In Vivo: Treatment with 1 mg/kg Maropitant citrate, significantly reduces the size of ulcerative dermatitis (UD) lesions in mice. Intravenous Maropitant decreases MAC by 16%. In contrast, epidural administration of either saline or Maropitant does not change the MAC (2.17% and 1.92 %, respectively).

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