基质金属蛋白酶-13(MMP-13)的药物drug discovery kit

基质金属蛋白酶-13(MMP-13)的药物drug disc

overy kit
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  • ¥6355
  • ENZO
  • USA
  • BML-AK413-0001
  • 2025年08月15日
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    • 详细信息
    • 技术资料
    • 英文名

      Matrix Metalloproteinase-13 (MMP-13) fluorometric drug discovery kit

    • 规格

      96wells

    基质金属蛋白酶-13(MMP-13)的药物drug discovery kit
    Matrix Metalloproteinase-13 (MMP-13) fluorometric drug discovery kit
    A QuantiZyme™ Assay System. The MMP-13 Fluorometric (also known as fluorimetric) Drug Discovery Kit is a complete assay system designed to screen inhibitors of matrix metalloproteinase-13 (MMP-13, collagenase-3) using a quenched fluorogenic peptide: OMNIMMP® fluorogenic substrate Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH. Mca fluorescence is quenched by the Dpa group until cleavage by MMPs at the Gly-Leu bond separates the two moieties. The assays are performed in a convenient 96-well microplate format. The kit is useful to screen inhibitors of MMP-13, a potential therapeutic target. Included are active enzyme, assay buffer, a prototypic control inhibitor (NNGH3), and a detailed instruction booklet.

    Product Specification

    Alternative Name: Collagenase-3
     
    Applications: Fluorescent detection, HTS
    Activity assay
     
    Shipping: Shipped on Dry Ice
     
    Long Term Storage: -80°C
     
    Kit/Set Contains: MMP-13 enzyme (human) (recombinant), substrate, calibration standard, inhibitor, assay buffer, 96-well white microplate.
     
    UniProt ID: P45452
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