For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -3090℃ for several months.
英文名:
EPZ5676
库存:
详询
供应商:
详询
CAS号:
1380288-87-8
规格:
2mg/5mg/10mg/25mg/50mg/1mL/10mM
规格:
2mg
产品价格:
¥680.0
规格:
5mg
产品价格:
¥1080.0
规格:
10mg
产品价格:
¥1730.0
规格:
25mg
产品价格:
¥3600.0
规格:
50mg
产品价格:
¥6300.0
规格:
1mL/10mM
产品价格:
¥980.0
ID:T3099
PURITY:0.98
Formula:C30H42N8O3
MolWt:562.71
Appearance:白色粉末
Solubility:G4DMSO:100 mg/mL warmed (177.71 mM)
Bioactivity:EPZ-5676 is an S-adenosyl methionine (SAM) competitive inhibitor of protein methyltransferase DOT1L with Ki of 80 pM, demonstrating >37,000-fold selectivity against all other PMTs tested, inhibits H3K79 methylation in tumor. Phase 1.