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- CAS号：
339539-92-3
- 规格：
25mg/50mg/100mg
| 规格： | 25mg | 产品价格： | ￥9360.0 |
|---|---|---|---|
| 规格： | 50mg | 产品价格： | ￥12240.0 |
| 规格： | 100mg | 产品价格： | ￥15600.0 |
Product Introduction
Bioactivity
| 名称 | Anamorelin Fumarate |
| 描述 | Anamorelin Fumarate is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay). |
| 体外活性 | No significant antagonist activity is observed with Anamorelin at concentrations of up to 1,000 nM. In the binding experiments, Anamorelin binds to the ghrelin receptor with a binding affinity constant (Ki) of 0.70 nM. In the competition assay with radiolabeled ibutamoren (another ghrelin receptor agonist), Anamorelin is also found to bind with high affinity to the ghrelin receptor (IC50: 0.69 nM). In rat pituitary cells incubated with Anamorelin, there is a dose-dependent stimulatory effect on GH release and the potency (EC50) is 1.5 nM. Anamorelin is screened for activity against a set of over 100 receptors, ion channels, transporters, and enzymes. Anamorelin demonstrates binding to the tachykinin neurokinin 2 (NK2) site (IC50: 0.021 μM); however, a subsequent NK2 functional assay demonstrates no functional activity. |
| 体内活性 | In rats, Anamorelin at an oral dose of 3, 10, or 30 mg/kg once daily significantly increases both food intake and body weight from Day 2 to Day 7 of treatment compared with the vehicle control. The cumulative change in food intake and weight gain increases dose-dependently, and these changes are significant at all dose levels compared to the control. Administration of Anamorelin at a single oral dose of 3, 10, or 30 mg/kg induces a dose-dependent increase in plasma GH levels and GH AUC0-6h in rats. |
| 存储条件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| 关键字 | RC-1291 Fumarate | RC 1291 Fumarate | ONO7643 Fumarate | ONO 7643 Fumarate | ghrelin receptor | Anamorelin Fumarate |
| 相关产品 | Obestatin (rat) acetate | Obestatin (human) | Anamorelin | Ibutamoren | CJC-1295 acetate(863288-34-0 free base) | Ibutamoren Mesylate | YIL 781 | AnaMorelin hydrochloride | Taurolithocholic Acid 3-sulfate sodium salt | L-692429 | Cortistatin-8 acetate | JMV 2959 hydrochloride (925238-89-7 free base) |
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非食品添加物指的是在食品生产过程中加入的非食品用化学物质，包括未经国务院卫生行政部门批准使用的添加剂和工业级（非食品级）原料。目前发现的一些非食品法添加物有：工业硫酸铜、酸性橙Ⅱ、富马酸二甲酯（DMF，克霉灵）、硼砂、荧光增白剂、苏丹红一号、孔雀石绿、吊白块、工业钛白粉、工业石蜡、结晶紫、工业淀粉、工业明胶、溴酸钾、工业漂白剂—漂白精、乌洛托品、铅铬绿、福尔马林、工业尿素、工业用盐等，还有一些非食品添加物在陆续发现。 目录 • 1. 工业
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富马酸阿拉莫林【339539-92-3】
￥9360 - 15600
