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- 详细信息
- 文献和实验
- 技术资料
- CAS号:
944997-60-8
- 规格:
1mg/5mg/10mg/25mg/50mg/100mg
| 规格: | 1mg | 产品价格: | ¥872.0 |
|---|---|---|---|
| 规格: | 5mg | 产品价格: | ¥2704.0 |
| 规格: | 10mg | 产品价格: | ¥3944.0 |
| 规格: | 25mg | 产品价格: | ¥6104.0 |
| 规格: | 50mg | 产品价格: | ¥7896.0 |
| 规格: | 100mg | 产品价格: | ¥11040.0 |
Product Introduction
Bioactivity
| 名称 | C3a Receptor Agonist |
| 描述 | C3a Receptor Agonist (C3a receptor agonist 1) binds the G protein-coupled C3a receptors (C3aRs) in the immune system complement pathway. Activation of C3aR prevents neutrophils from being mobilized in a model of intestinal ischemia-reperfusion injury. C3aRs are expressed on neural progenitor cells and immature neurons in adult mice. C3a stimulates differentiation of neural progenitor cells in vitro. |
| 存储条件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| 溶解度 | DMF : 30 mg/mL (69.19 mM), Sonication is recommended. DMSO : 40 mg/mL (92.25 mM), Sonication is recommended. Ethanol : 30 mg/mL (69.19 mM), Sonication is recommended. |
| 关键字 | ComplementSystem | Complement System | C3a Receptor Agonist | C3a |
| 相关产品 | Cyclosporin A | Dexamethasone acetate | CP-289 | Dextran sulfate sodium salt (MW 5000) | Dexamethasone | BCX 1470 hydrochloride | Iptacopan hydrochloride | ADH-503 | Iptacopan | 3-Phenoxybenzaldehyde | EG01377 2HCl | Avacopan |
| 相关库 | Bioactive Compound Library | Bioactive Compounds Library Max | Immunology/Inflammation Compound Library |
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文献和实验Filtration 1. Sample: 5–10 mL pooled Wnt3A-containing fractions fromSection 2.3.2 . 2. HiLoad 26/60 Superdex 200 preparative grade. 3. Buffer: 1× PBS, 1% (w/v) CHAPS. 4. Syringe (30 mL) with 0.2-μm pore size filter. 2.3.4. Step 4: Heparin
β-受体激动剂是一类苯乙醇胺类化合物,在动物体内能减缓或减少脂肪沉积,增加肌肉蛋白沉淀,提高动物胴体瘦肉率、增重和提高饲料转化率,当用于牛、羊、禽、猪等畜禽的促生长剂、饲料添加剂时,会提高其瘦肉率,但同时,β-受体激动剂类药物也可引起心室早搏,四肢、脸、颈部骨骼肌震颤,还引发代谢紊乱,对糖尿病人可发生酸中毒或酮中毒。由于其严重的危害性,在许多国家包括欧盟和中国已禁止在饲料中添加这些化合物,相关标准规定需对动物源性食品、饲料、饮用水中该类化合物的残留量进行检测。β-受体激动剂类药物进入人或动物
,无效或症状加重可改用或并用左旋多巴。 2.中期病人可服用美多巴或倍尼美。 3.晚期或重症病人在(2)基础上可加用受体激动剂如溴隐停等。 4.身体状况好,以单侧震颤为主,且非主侧(右利手的左半身),及用药治疗无效,可考虑手术治疗(X刀等定向治疗)。 辅助检查 1.对诊断明确者检查基本上以检查框限“A”为主。 2.对起病年龄较轻或诊断不明需与震颤麻痹综合征(继发性震颤麻痹)鉴别,检查专案可包括检查框限“A”、“B”、“C”。 疗效评价 1.治愈:症状体征消失
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