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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
零下80~20°C
- 保质期:
Powder: -20°C for 3 years In solvent: -80°C for 2 years
- 英文名:
Estrogen receptor β antagonist 2
- 库存:
10
- 供应商:
TargetMol
- CAS号:
2580941-14-4
- 规格:
100 mg/50 mg/25 mg
| 规格: | 100 mg | 产品价格: | ¥17500.0 |
|---|---|---|---|
| 规格: | 50 mg | 产品价格: | ¥13800.0 |
| 规格: | 25 mg | 产品价格: | ¥10600.0 |
Product Introduction
Bioactivity
英文名:Estrogen receptor β antagonist 2
描述:Estrogen receptor β antagonist 2 is a selective, potent estrogen receptor β (ERβ) antagonist that acts on Erα (IC50: 109.10 μM) and Erβ (IC50: 0.63 μM).

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文献和实验Cotransfection Assays and Steroid Receptor Biology
The glucocorticoid, mineralocorticoid, progesterone, androgen, estrogen α and estrogen β receptors (GR, MR, PR, AR, ERα, and ERβ, respectively) form the steroid receptor family, part of the nuclear receptor superfamily
Overview of Receptor Allosterism
Figure 1.21.2 Effect of: (A ) negative allosteric modulator, (B ) positive allosteric modulator, or (C ) a competitive antagonist on orthosteric ligand‐receptor occupancy (ρA ). For all the simulations, p K
Characterization of Nuclear Receptor Ligands by Multiplexed Peptide Interactions
, although described for nuclear receptors, may also be applied to other types of molecular interactions. Keywords: Microsphere; flow cytometry; nuclear receptor; coactivator; corepressor; cofactor; agonist; antagonist; ligand; ligand binding
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