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- 2025年12月05日
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- 详细信息
- 文献和实验
- 技术资料
- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
2580941-14-4
- 规格：
5 mg/10 mg
| 规格： | 5 mg | 产品价格： | ￥2800.0 |
|---|---|---|---|
| 规格： | 10 mg | 产品价格： | ￥4500.0 |
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Estrogen receptor β antagonist 2
CAS No. : 2580941-14-4
MCE 国际站：Estrogen receptor β antagonist 2
产品活性：Estrogen receptor β antagonist 2 是一种有效的选择性雌激素受体β estrogen receptor β (ERβ) 拮抗剂，对 Erα 和 Erβ 的 IC50 值为 109.10，0.63 µM。
研究领域：Vitamin D Related/Nuclear Receptor
作用靶点：Estrogen Receptor/ERR
In Vitro: Estrogen receptor β antagonist 2 (compound 42) (0-100 µM) shows antiproliferative activity with IC50 value of >100 µM in MCF-7cells.
.Estrogen receptor β antagonist 2 exhibits differences in interaction potential to H12 of ERβ via Asp303 (H3) H-bonding to Tyr488.
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