LPA5 antagonist 2,2839471-44-0

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LPA5 antagonist 2

CAS No. : 2839471-44-0

MCE 国际站：LPA5 antagonist 2

产品活性：LPA5 antagonist 2 (compound 65) 是高水溶性的 LPA5 (lysophosphatidic acid receptor 5) 拮抗剂。LPA5 antagonist 2 显著减轻痛觉，可用于炎症性和神经性疼痛的研究。

研究领域：Others

作用靶点：Others

In Vitro: LPA5 antagonist 2 (0-10 μM) inhibits hLPA5 calcium mobilization with an IC₅₀ value of 69 nM and inhibits hLPA5 cAMP with an IC₅₀ value of 340 nM.
LPA5 antagonist 2 (0-10 μM) shows no significant affinity for other receptors, exhibits good target selectivity for LPA5.

In Vivo: LPA5 antagonist 2 (5.3-17.8 mg/kg; i.p. once) alleviates CFA-induced inflammatory pain in vivo.

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