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- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥2105.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥940.0 |
| 规格: | 5 mg | 产品价格: | ¥2000.0 |
| 规格: | 10 mg | 产品价格: | ¥3200.0 |
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AZD1656
CAS No. : 919783-22-5
MCE 国际站:AZD1656
产品活性:AZD1656 是一种有效的,选择性的,具有口服活性的葡萄糖激酶 (glucokinase) 激活剂,EC50为 60 nM,可用于 2 型糖尿病的研究。
研究领域:Metabolic Enzyme/Protease
作用靶点:Glucokinase
In Vivo: AZD1656 (0-9 mg/kg; oral gavage; daily; for 8 weeks; C57BL/6 mice) treatment shows lowered blood glucose and glucose excursion and raised insulin. Liver mRNA levels for various ChREBP target genes including carbohydrate response element binding protein beta isoform (ChREBP-β), G6pc, Pklr, Acly, Acac and Gpd2 are increased by AZD1656.
相关产品:Drug Repurposing Compound Library Plus | Clinical Compound Library Plus | Bioactive Compound Library Plus | Kinase Inhibitor Library | Metabolism/Protease Compound Library | Clinical Compound Library | Drug Repurposing Compound Library | Anti-diabetic Compound Library | Glycolysis Compound Library | Orally Active Compound Library | Anti-Cancer Metabolism Compound Library | Glucose Metabolism Compound Library | Targeted Diversity Library | Highly Selective Activators Library | Dorzagliatin | Palmitelaidic Acid | RO-28-1675 | MK-0941 | GKA50 | Globalagliatin | AMG-3969 | Nerigliatin | AR453588 | PF-04991532 | AM-2394 | BMS-820132 | Glucokinase activator 3 | IHVR-11029 | AMG-1694 | AZD1092 | Cadisegliatin | CM-10-18 | Glucokinase activator 6 | Glucokinase activator 1 | PSN-GK1
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0126 ★ 白介素-2(IL-2) ELISA 48T/96T 1000/1800 进口分装 F0127 可溶性白介素-2 受体 (sIL-2R) ELISA 48T/96T 1000/1800 进口分装 F0128 白介素-3(IL-3) ELISA 48T/96T 1000/1800 进口分装 F0129 ★ 白介素-4(IL-4) ELISA 48T/96T 1000/1800 进口分装 F0130 白介素-5(IL-5
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