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- 详细信息
- 技术资料
- 保存条件:
4°C, sealed storage, away from moisture and light
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1217195-61-3
- 规格:
1 mg/5 mg/10 mg/25 mg/50 mg/100 mg
| 规格: | 1 mg | 产品价格: | ¥290.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥640.0 |
| 规格: | 10 mg | 产品价格: | ¥1000.0 |
| 规格: | 25 mg | 产品价格: | ¥2000.0 |
| 规格: | 50 mg | 产品价格: | ¥3000.0 |
| 规格: | 100 mg | 产品价格: | ¥4500.0 |
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CP-31398 dihydrochloride
CAS No. : 1217195-61-3
MCE 国际站:CP-31398 dihydrochloride
产品活性:CP-31398 dihydrochloride 在 p53 突变或野生型的癌细胞中,稳定 p53 的活性构象、促进 p53 的活性。
研究领域:Apoptosis
作用靶点:MDM-2/p53
In Vitro: CP-31398 (36.75 μM, 16 h) induces p21 in p53-mutant cells.
CP-31398 (15 μg/mL, 20 hours) could induce apoptosis and cell cycle arrest in SW480 cells.
In Vivo: CP-31398 (100 mg/kg, orally) exhibits significant anti-tumor activity in mice models.
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