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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1312815-93-2
- 规格:
1 mg/5 mg
| 规格: | 1 mg | 产品价格: | ¥1845.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥4612.0 |
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PF-4693627
CAS No. : 1312815-93-2
MCE 国际站:PF-4693627
产品活性:PF-4693627 是一种有效的,口服生物可利用的,选择性的微粒体前列腺素E合酶 (mPGES-1) 抑制剂 (IC50=3 nM),可用于骨关节炎和类风湿关节炎等的研究。
作用靶点:PGE synthase
In Vitro: PF-4693627 also inhibits mPGES-1 with IC50s of 180 and 6 nM in HWB-1483 and human fetal fibroblast, respectively.
PF-4693627 shows high activity in lipopolysaccharide (LPS) stimulated human whole blood (HWB) cell assay (IC50=109 nM).
In Vivo: PF-4693627 (10 mg/kg; orally) inhibits 63% of PGE2 production relative to vehicle control in Guinea pig carrageenan stimulated air pouch model.
PF-4693627 (1.0 mg/kg; i.v.) shows good bioavailability (59%) and modest half life (t1/2=3.7 h) in Sprague-Dawley rats.
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文献和实验字(0x93)。读取坐标值的C程序如下: intTouch_GetXY() {…… for(i=;i {rPDATG|=0x40;/*DCLK为高*/ temp=(rPDATF>>7); temp&=0x1;/*通过PF7逐位读取坐标值*/ data|=temp Delay(220);/*delay220ns*/ rPDATG&=0xBF;/*DCLK为低*/ Delay(220
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