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- 2025年12月05日
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- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
1639220-19-1
- 规格：
1 mg/5 mg/10 mg/25 mg
| 规格： | 1 mg | 产品价格： | ￥703.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥1863.0 |
| 规格： | 10 mg | 产品价格： | ￥2988.0 |
| 规格： | 25 mg | 产品价格： | ￥4788.0 |
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Sigma-1 receptor antagonist 1
CAS No. : 1639220-19-1
MCE 国际站：Sigma-1 receptor antagonist 1
产品活性：Sigma 1 receptor antagonist 1 (compound 137) 是一种高效选择性的 sigma-1 受体 (σ1R) 拮抗剂，对 σ1R 具有高亲和力 (Ki = 1.06 nM)。Sigma 1 receptor antagonist 1 具有抗神经痛活性，有作为研究神经性疼痛活性分子的前景。
研究领域：Neuronal Signaling
作用靶点：Sigma Receptor
In Vitro: Sigma?1 receptor antagonist 1 exhibits a high binding affinity to σ1R receptor (Ki = 1.06 nM) and good σ-1/2 selectivity (1344-fold).
In Vivo: Sigma?1 receptor antagonist 1 exerts dose-dependent antinociceptive effects in mice formalin model and rats CCI models of neuropathic pain.
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