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- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1024448-59-6
- 规格:
10 mM * 1 mL/5 mg/10 mg/25 mg/50 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥770.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥700.0 |
| 规格: | 10 mg | 产品价格: | ¥1300.0 |
| 规格: | 25 mg | 产品价格: | ¥2600.0 |
| 规格: | 50 mg | 产品价格: | ¥4700.0 |
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RN-1747
CAS No. : 1024448-59-6
MCE 国际站:RN-1747
产品活性:RN-1747 是选择性的瞬时受体电位阳离子通道 V 型亚家族成员4 (TRPV 4) 的激动剂,其对hTRPV4、mTRPV4 和rTRPV4 的EC50 值分别为0.77 μM、4.0 μM 和4.1 μM。RN-1747 还能拮抗TRPM8,其IC50 值为4.0 μM。
研究领域:Membrane Transporter/Ion Channel | Neuronal Signaling
作用靶点:TRP Channel
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