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- 详细信息
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
K03861
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
853299-07-7
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥1324.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥457.0 |
| 规格: | 5 mg | 产品价格: | ¥1200.0 |
| 规格: | 10 mg | 产品价格: | ¥1400.0 |
| 规格: | 25 mg | 产品价格: | ¥2940.0 |
| 规格: | 50 mg | 产品价格: | ¥4700.0 |
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AUZ 454
CAS No. : 853299-07-7
MCE 国际站:AUZ 454
产品活性:AUZ 454 (K03861) 是一个 type II CDK2 的抑制剂,Kd 值是 8.2 nM。
研究领域:Cell Cycle/DNA Damage
作用靶点:CDK
In Vitro: AUZ 454 (K03861) (10-20 μM; 1, 2, 3, and 4 days) has a inhibitory effect on Caki-1 and ACHN cells with WTAP overexpression by CCK8 assays.
AUZ 454 (K03861) (10 μM; 24 hours) decreases the colony fold in Caki-1 and ACHN cells through a CDK2-dependent mechanism.
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