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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1609389-52-7
- 规格:
10 mM * 1 mL/10 mg/25 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥4180.0 |
|---|---|---|---|
| 规格: | 10 mg | 产品价格: | ¥3800.0 |
| 规格: | 25 mg | 产品价格: | ¥5800.0 |
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ACY-957
CAS No. : 1609389-52-7
MCE 国际站:ACY-957
产品活性:ACY-957 是一种具有口服活性,选择性的 HDAC1 和 HDAC2 抑制剂,对 HDAC1/2/3 的 IC50 值分别为 7 nM,18 nM 和 1300 nM,对 HDAC4/5/6/7/8/9 无作用。
研究领域:Cell Cycle/DNA Damage | Epigenetics
作用靶点:HDAC
In Vitro: ACY-957 is a selective inhibitor of HDAC1 and HDAC2, with IC50s of 7 nM, 18 nM, and 1300 nM against HDAC1/2/3, respectively, and shows no inhibition on HDAC4/5/6/7/8/9. ACY-957 has an IC50 of 304 nM for HDAC2 in primary hematopoietic progenitors.
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