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- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
848217-00-5
- 规格：
10 mM * 1 mL/5 mg/10 mg/50 mg/100 mg
| 规格： | 10 mM * 1 mL | 产品价格： | ￥825.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥750.0 |
| 规格： | 10 mg | 产品价格： | ￥1150.0 |
| 规格： | 50 mg | 产品价格： | ￥3900.0 |
| 规格： | 100 mg | 产品价格： | ￥5600.0 |
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H4 Receptor antagonist 1
CAS No. : 848217-00-5
MCE 国际站：H4 Receptor antagonist 1
产品活性：H4 Receptor antagonist 1 是一种有效的、有选择性的组胺H4受体 (H4R) 的反向激动剂，其IC50 值为19 nM。
研究领域：GPCR/G Protein | Neuronal Signaling | Immunology/Inflammation
作用靶点：Histamine Receptor
In Vitro: H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
In Vivo: H4 Receptor antagonist 1 indicates that metabolic stability in rat microsomes is very low with only 1% parent compound remaining after 10 min incubation.
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