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- 详细信息
- 文献和实验
- 技术资料
- 库存:
97
- 英文名:
SCH-1473759 hydrochloride
- CAS号:
1094067-13-6
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|2mg|5mg|10mg|50mg|100mg
特别提示:包括Aurora A和Aurora B抑制剂(SCH-1473759 hydrochloride)在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:Aurora A和Aurora B抑制剂(SCH-1473759 hydrochloride)
英文名称:SCH-1473759 hydrochloride
产品货号:M01797
产品规格:1mL(10mM)|2mg|5mg|10mg|50mg|100mg
SCH1473759盐酸盐是Aurora A和Aurora B高效抑制剂,IC50值分别为4nM和13nM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:1094067-13-6
纯度:99.06%
分子式:C₂₀H₂₇ClN₈OS
分子量:463.0
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
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文献和实验A method for analyzing the ubiquitination and degradation of aurora-A
has been well characterized and it was shown that it is ubiquitin proteasome pathway that leads to the elimination of cyclins. By now, many other regulatory proteins were shown to be degraded by the same pathway, among them members of the aurora kinase family, degraded
Studying the Roles of Aurora-C Kinase During Meiosis in Mouse Oocytes
We previously isolated Aurora-C (Aurkc/Aie1 ) in a screen for kinases expressed in mouse sperm and eggs. Aurora-C kinase was reported to be a chromosomal passenger protein that plays critical roles in chromosome alignment
The Ipl1/Aurora Kinase Family: Methods of Inhibition and Functional Analysis in Mammalian Cells
and the pharmaceutical industry. Indeed, two small molecule Aurora kinase inhibitors have recently been described. In this chapter, we describe several methods for investigating the function of the Aurora kinases, focusing on Aurora B. We describe the use of the small
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