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- 详细信息
- 文献和实验
- 技术资料
- 库存:
91
- 英文名:
GW0742
- CAS号:
317318-84-6
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|5mg|10mg|50mg|100mg
特别提示:包括高度PPARδ激动剂(GW0742)在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:高度PPARδ激动剂(GW0742)
英文名称:GW0742
产品货号:M00560
产品规格:1mL(10mM)|5mg|10mg|50mg|100mg
GW0742(GW610742)是一种有效的高度选择性PPARδ激动剂,作用于PPARδ,-α,和-γ受体,EC50值分别为1nM,1.1μM and2μM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:317318-84-6
别名:GW610742
纯度:99.63%
分子式:C₂₁H₁₇F₄NO₃S₂
分子量:471.49
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
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文献和实验at all the conditions? 2, if the positive control turns out the predict result, it's possible your drug may exert its anti-inflamation effect not through the reported PPAR pathway. and GW9662 can potentiate the other anti-inflamation pathway. So you may want
. A new drug candidate belonging to the family of the peroxisome proliferator-activated receptor-delta agonists termed GW1516 (also referred to as GW501516) has been prohibited by the World Anti-Doping Agency in 2009
PPAR/ Agonist Increases the Expression of PGE2 Receptor Subtype EP4 in Human Lung Carcinoma Cells
and that treatment with a selective PPARβ/δ agonist, GW501516, stimulated the expression of EP4 and induced NSCLC cell proliferation. In addition, this PPARβ/δ agonist also induced EP4 promoter activity through the binding of C/EBP to the NF-IL6 site in the EP
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