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- 详细信息
- 文献和实验
- 技术资料
- 库存:
419
- 英文名:
FIPI
- CAS号:
939055-18-2
- 保质期:
2年
- 供应商:
北京百奥莱博科技有限公司
- 保存条件:
-20℃,有效期2年,溶入溶剂后-20℃
- 规格:
1mL(10mM)|5mg|10mg|50mg|100mg
特别提示:包括PLD1和PLD2抑制剂(FIPI)在内,本公司的所有产品仅可用于科研实验,严禁用于临床医疗及其他非科研用途!
产品名称:PLD1和PLD2抑制剂(FIPI)
英文名称:FIPI
产品货号:M04492
产品规格:1mL(10mM)|5mg|10mg|50mg|100mg
FIPI是halopemide的衍生物,能够有效抑制PLD1和PLD2,IC50值分别为25nM和20nM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:939055-18-2
别名:5-Fluoro-2-indolyl deschlorohalopemide
纯度:99.53%
分子式:C₂₃H₂₄FN₅O₂
分子量:421.47
结构式:
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
除了PLD1和PLD2抑制剂(FIPI),5-Fluoro-2-indolyl deschlorohalopemide,我公司还供应以下相关产品:
KFS286 细胞衰老检测试剂盒(β-半乳糖苷酶检测试剂盒) 100T
M00272 PI3K/mTOR/DNA-PK抑制剂(LY3023414) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M00515 MMPs抑制剂(Marimastat) 1mL(10mM)|1mg|5mg|10mg|50mg
M00667 JAK2抑制剂(CHZ868) 1mL(10mM)|2mg|5mg|10mg|25mg|50mg|100mg
M00707 BET蛋白抑制剂(GSK1324726A) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M00732 Aurora A和Aurora B抑制剂(ZM447439) 1mL(10mM)|5mg|10mg|50mg
M00962 FAK和ALK双重抑制剂(CEP-37440) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M01156 AGC kinase抑制剂(AT13148) 1mL(10mM)|5mg|10mg|50mg|100mg
M01187 c-Abl激活剂(DPH) 1mL(10mM)|10mg|50mg
M01300 肽酶抑制剂(NSC632839) 1mL(10mM)|5mg|10mg|25mg|50mg|100mg
M01419 EZH2抑制剂(CPI-169 racemate) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M01625 VEGFR2抑制剂(Cediranib maleate) 1mL(10mM)|5mg|10mg|50mg|100mg
M01640 Aurora A和B抑制剂(CYC-116) 1mL(10mM)|5mg|10mg|50mg|100mg
M02240 苯二氮逆转激动剂(DMCM hydrochloride) 1mL(10mM)|5mg|10mg|25mg|50mg|100mg
M02277 HDAC抑制剂(PTACH) 1mL(10mM)|5mg|10mg|50mg
M02789 NEP抑制剂(AHU-377) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M04046 壳聚糖酶和乙酰氨基己糖苷酶抑制剂(Chitinase-IN-1) 1mL(10mM)|2mg|5mg|10mg|50mg|100mg
M04232 脂质过氧化抑制剂(Eugenol) 1mL(10mM)|100mg|500mg
M04378 JAK1抑制剂(Upadacitinib) 1mL(10mM)|1mg|5mg|10mg|25mg
M04412 JAK3抑制剂(Decernotinib) 1mL(10mM)|2mg|5mg|10mg|25mg|50mg
M04489 前列腺素合成抑制剂(Sulindac) 1mL(10mM)|100mg|500mg
M04490 组胺N-甲基转移酶抑制剂 1mL(10mM)|100mg
M05273 DPP-4抑制剂(Linagliptin) 1mL(10mM)|5mg|10mg|50mg|100mg|250mg
M06034 肾上腺*受体抑制剂 1mL(10mM)|10mg|50mg|100mg
M06405 mAChR激动剂 1mL(10mM)|1mg|5mg
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文献和实验Assay of Phospholipase D Activity in Cell-Free Systems
. The two mammalian PLD isoforms, PLD1 and PLD2, are peripheral membrane proteins that exhibit important physical and functional interactions with the actin cytoskeleton. We outline a cell-free system for the characterization of mammalian PLDs and their activation
Reconstitution System Based on Cytosol-Depleted Cells to Study the Regulation of Phospholipase D
Phospholipase D (PLD) hydrolyzes phosphatidylcholine to produce the membraneassociated second messenger, phosphatidic acid (PA) and choline. Two phospholipase D enzymes—PLD1 and PLD2—have been identified, although their regulatory mechanisms
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