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- 2025年12月04日
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- 详细信息
- 询价记录
- 技术资料
- 保存条件：
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名：
SCH 530348
- 库存：
货期：1-2天
- 供应商：
MedChemExpress LLC
- CAS号：
618385-01-6
- 规格：
10 mM * 1 mL/1 mg/5 mg/10 mg/25 mg/50 mg
| 规格： | 10 mM * 1 mL | 产品价格： | ￥1296.0 |
|---|---|---|---|
| 规格： | 1 mg | 产品价格： | ￥598.0 |
| 规格： | 5 mg | 产品价格： | ￥1196.0 |
| 规格： | 10 mg | 产品价格： | ￥1913.0 |
| 规格： | 25 mg | 产品价格： | ￥3461.0 |
| 规格： | 50 mg | 产品价格： | ￥5191.0 |
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Vorapaxar
CAS No. : 618385-01-6
MCE 国际站：Vorapaxar
产品活性：Vorapaxar (SCH 530348)，抗血小板活性分子，是一种选择性、口服活性和竞争性的凝血酶受体蛋白酶激活受体 (PAR-1) 拮抗剂，Ki 值为 8.1 nM。Vorapaxar (SCH 530348) 剂量依赖性抑制凝血酶受体激活肽 (TRAP) 诱导的血小板聚集。
研究领域：GPCR/G Protein
作用靶点：Protease Activated Receptor (PAR)
In Vitro: Vorapaxar (SCH 530348) shows potent inhibition of thrombin-induced platelet aggregation with an IC50 of 47 nM and haTRAP-induced platelet aggregation with an IC50 of 25 nM. Vorapaxar (SCH 530348) inhibits thrombininduced calcium transient in human coronary artery smooth muscle cells (HCASMC) with a Ki of 1.1 nM. It also inhibits thrombin-stimulated thymidine incorporation in HCASMC with a Ki of 13 nM.
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