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- 文献和实验
- 技术资料
- 保存条件:
零下80~20°C
- 保质期:
Powder: -20°C for 3 years In solvent: -80°C for 2 years
- 英文名:
LGK974
- 库存:
10
- 供应商:
TargetMol
- CAS号:
1243244-14-5
- 规格:
1 mL/5 mg/25 mg/100 mg/1 mg/50 mg/2 mg/10 mg
| 规格: | 1 mL | 产品价格: | ¥941.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥997.0 |
| 规格: | 25 mg | 产品价格: | ¥3210.0 |
| 规格: | 100 mg | 产品价格: | ¥6680.0 |
| 规格: | 1 mg | 产品价格: | ¥438.0 |
| 规格: | 50 mg | 产品价格: | ¥4680.0 |
| 规格: | 2 mg | 产品价格: | ¥632.0 |
| 规格: | 10 mg | 产品价格: | ¥1790.0 |
Product Introduction
Bioactivity
英文名:LGK974
描述:LGK974 (NVP-LGK974) is an effective and selective PORCN inhibitor and inhibits Wnt signaling (IC50: 0.4 nM) in TM3 cells. It has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

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文献和实验Wnt与Hedgehog:两条"平行"通路,信号运行逻辑竟不谋而合?
mAb (S-2678-117) 抗体 2915 Wnt Signaling Antibody Sampler Kit 抗体套装 S0M1069 Wnt/β-Catenin Signaling Pathway Antibody MiniAb Set 抗体套装 26118 Hedgehog Signaling Antibody Sampler Kit 抗体套装 abs811224 LGK974 Wnt抑制剂 abs810648 XAV-939 Wnt抑制剂 abs812230
1.000 1.000 1.000 2 0.500 0.800 0.900 0.950 0.980 0.990 0.995 0.998 0.999 3 0.404 0.687 0.805 0.878 0.934 0.959 0.974 0.986 0.991 4 0.347 0.603 0.729 0.811 0.882 0.917 0.942 0.963 0.974 5 0.309 0.551 0.669 0.755 0.833 0.875 0.906 0.935 0.951 6 0.281
, A., et al., Switchable photooxygenation catalysts that sense higher-order amyloid structures. Nature Chemistry, 2016. 8(10): p. 974-982.3.Ni, J., et al., Near-Infrared Photoactivatable Oxygenation Catalysts of Amyloid Peptide. Chem, 2018. 4(4): p. 807-820
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