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- 文献和实验
- 技术资料
- 保存条件:
详询
- 保质期:
12 months from date of receipt.
- 英文名:
EGFR/HER2/DHFR-IN-3
- 库存:
99
- 供应商:
Biorbyt
- 规格:
5 mg/50 mg
| 规格: | 5 mg | 产品价格: | ¥0.0 |
|---|---|---|---|
| 规格: | 50 mg | 产品价格: | ¥0.0 |
类别: Small Molecules
描述: EGFR/HER2/DHFR-IN-3 is a potent dual inhibitor of EGFR (IC50=0.138 µM) and HER2 (IC50=0.092 µM), with additional DHFR inhibition (IC50=0.193 µM). It induces S-phase cell cycle arrest and apoptosis in MCF7 breast cancer cells, supporting its application in oncology research and mechanistic studies.
靶点: EGFR,Apoptosis,DHFR
研究领域: Cardiovascular Research, Cell Biology, Metabolism Research, Metabolism Research; Cell Biology, Molecular Biology, Signal Transduction
保存条件: -20°C
备注: For research use only.
描述: EGFR/HER2/DHFR-IN-3 is a potent dual inhibitor of EGFR (IC50=0.138 µM) and HER2 (IC50=0.092 µM), with additional DHFR inhibition (IC50=0.193 µM). It induces S-phase cell cycle arrest and apoptosis in MCF7 breast cancer cells, supporting its application in oncology research and mechanistic studies.
靶点: EGFR,Apoptosis,DHFR
研究领域: Cardiovascular Research, Cell Biology, Metabolism Research, Metabolism Research; Cell Biology, Molecular Biology, Signal Transduction
保存条件: -20°C
备注: For research use only.
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EGFR/HER2/DHFR-IN-3,orb1942274,Biorbyt
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