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货期：1-2天
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- CAS号：
1204572-55-3
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1 mg/5 mg/10 mg/25 mg/50 mg/100 mg
| 规格： | 1 mg | 产品价格： | ￥234.0 |
|---|---|---|---|
| 规格： | 5 mg | 产品价格： | ￥654.0 |
| 规格： | 10 mg | 产品价格： | ￥1041.0 |
| 规格： | 25 mg | 产品价格： | ￥2225.0 |
| 规格： | 50 mg | 产品价格： | ￥3288.0 |
| 规格： | 100 mg | 产品价格： | ￥4700.0 |
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BPAM344
CAS No. : 1204572-55-3
MCE 国际站：BPAM344
产品活性：BPAM344 是红藻氨酸受体 (KAR) 亚基 GluK1b、GluK2a 和 GluK3a 的正变构调节剂 (PAM)。
研究领域：Membrane Transporter/Ion Channel | Neuronal Signaling
作用靶点：iGluR
In Vitro: BPAM344 potentiates glutamate-evoked currents of GluK2a 21-fold at the highest concentration tested (200 μM), with an EC50 of 79 μM. BPAM344 markedly decreases desensitization kinetics (from 5.5 to 775 ms), whereas it only has a minor effect on deactivation kinetics.
BPAM344 (100 μM) also potentiates the peak current amplitude of KAR subunits GluK3a (59-fold), GluK2a (15-fold), GluK1b (5-fold), as well as the AMPA receptor subunit GluA1i (5-fold).
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文献和实验Pheromone Halo Assay REFERENCE: Hoffman, G., Garrison, T. R., and Dohlman, H. G., Analysis of RGS proteins in Saccharomyces cerevisiae , Methods Enzymol. 344:617-631, 2002. -Use sterile technique and sterile
3 二氢苊 254.33 254.33 254.42 254.36 254.39 254.44 4 芴 270.20 270.26 270.26 270.24 270.31 270.26 5 菲 300.00 300.00 300.00 300.00 300.00 300.00 6 蒽 301.5 301.59 301.57 301.55 301.55 301.50 7 荧蒽 344.73 344.67 344.77 344.78 344.76 344.74 8 芘 352
receptor was quantified by measuring the initial rate of substrate hydrolysis at 405 nm and same amount of proteins was used in the binding assays. Gray, T. E., Eisenstein, M., Yayon, A. and Givol, D. (1996). Asparagine-344 Is a Key Residue For Ligand
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