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CM10
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Powder: -20°C, 3 years; 4°C, 2 years. In solvent: -80°C, 6 months; -20°C, 1 month.
货期:1-2天
MedChemExpress LLC
10 mM * 1 mL/5 mg/10 mg/25 mg/50 mg/100 mg
MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
CAS No. : 692269-09-3
MCE 国际站:CM10
产品活性:CM10 是一种有效的,选择性乙醛脱氢酶 1A (ALDH1A) 家族抑制剂,对于 ALDH1A1,ALDH1A2 和 ALDH1A3 的 IC50 分别为 1700、740 和 640 nM。CM10 对 ALDH 家族其他成员没有抑制作用。CM10 可以调节新陈代谢并具有抗癌活性。
研究领域:Metabolic Enzyme/Protease
作用靶点:Aldehyde Dehydrogenase (ALDH)
In Vitro: CM10 (12.5, 25, 50, 100 μM; 1 hour) inhibits ALDEFLUOR activity in live cells and preferentially depletes CD133+ ovarian cancer stem-like cells (CSCs). ?CM10 induces a cellular/nuclear swelling necroptotic phenotype.
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