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- 详细信息
- 文献和实验
- 技术资料
- 库存:
52
- 英文名:
SCH-1473759 hydrochloride
- 保质期:
详见说明书
- 供应商:
上海一研
- 保存条件:
低温
- 规格:
1mL(10mM)|2mg|5mg|10mg|50mg|100mg
英文名称:SCH-1473759 hydrochloride
产品规格:1mL(10mM)|2mg|5mg|10mg|50mg|100mg
发货周期:1~3天
SCH1473759盐酸盐是Aurora A和Aurora B高效抑制剂,IC50值分别为4nM和13nM。
注:本品仅可用于科研实验,严禁用于临床医疗及其他用途!
CAS号:1094067-13-6
纯度:99.06%
分子量:463.0
储存条件:-20℃,有效期2年,溶入溶剂后-20℃请尽量在一个月内使用。
以下是细胞生物学试剂的详细介绍:
Aurora A和Aurora B抑制剂(SCH-1473759 hydrochloride) 细胞生物学研究有以下几个方面:
细胞生物学的研究内容十分广泛,主要包括:
①细胞核、染色体以及基因表达的研究;
②生物膜与细胞器的研究;
③细胞骨架体系的研究;
④细胞增殖及其调控;
⑤细胞分化及其调控;
⑥细胞的衰老与编程性死亡(凋亡);
⑦细胞的起源与进化;
⑧细胞工程.
细胞生物学研究的常用技术有哪些:
1.显微技术:包括显微观察,显微操作.
2细胞组分分析技术:离心分离技术,生物大分子定位技术,定量细胞化学分析技术.
3.细胞工程:细胞培养。
注意事项:
1. 本试剂盒的检测试剂中含有萤光素酶,反复冻融会导致其逐渐失活。尽管经测试本试剂反复冻融5次对于其检测效果无显著影响,为取得良好的使用效果,*次解冻后可适当分装保存。反复冻融过程中,可能会导致检测试剂中出现少量沉淀,此时宜平衡至室温,并尽量溶解。如仍有残留的不溶物,可以离心去除后使用,经测试不会影响后续的检测效果。
2. 检测时需使用白色或黑色的96孔板或384孔板。如果使用普通透明的96孔板或384孔板,相邻孔之间会产生相互干扰。
3. 使用说明中提供了检测ATP标准品的方法,实际检测细胞活力时通常并不需要检测ATP标准品。
cyclic GMP3',5'-环一磷鸟苷盐500u高纯,
Cyclo-C盐环胞5克试剂级,99%
Cyclohexanol六100克GR,99.8%
Cyclohexanone环已25克AR,99.8%
Cyclooctanone环辛25克BR,97%
Cyclopentanol羟基环500克AR,99%
Cyclopentanone oxime环肟100毫克CP,
Cyclosporin A环孢霉素A100毫克BR,2ml/支
CyDTA反-1,2-环己二-N,N,N',N'-四25克BR,97%,油状
Cys-GlyH-半胱-甘-OH100克BR,
Cytidine胞嘧核苷7.5KUBR,
Cytisine野靛碱5克BR
Cytochalasin B松胞菌素B1公斤BR,600u/mg,猪胰
Cytochrome C细胞血素C100克BR,0.5u/mg
Cytosine4-基-2-羟基嘧250UBR,99%
N-氧基匹格列酮 质量规格:>98%,BR NDSB 256
N-氧基帕潘立酮 质量规格:BR NDSB-211
N-氧基帕洛诺司琼 质量规格:Ind Grade Neutral red solution(1X)
N-氧基喹平 质量规格:>99.5%,SP Nickel powder
N-氧基奥平 质量规格:>65%,BS Nile blue A
N-亚硝基-N-基尿烷(>95.0%(GC)) 质量规格:>98%,BR N-Iodosuccinimide
N-溴代二酰亚(NBS) 质量规格:>99%,BR N-N-Dimethylglycine hydrochloride
N-辛酰基-N-基葡糖(MEGA-8) 质量规格:>98%,BC n-Nonyl-beta-D-maltopyranoside
n-辛基-β-D-吡喃葡萄糖苷(OGP) 质量规格:>98% (HPLC),BC n-Octyl-b-D-maltopyranoside
N-硝基-L-精氨酸酯 质量规格:>98%,BC Nonyl β-D-glucopyranoside
Aurora A和Aurora B抑制剂(SCH-1473759 hydrochloride) 吲达帕 Indapamide 26807658 规格:>99%,EP6.0,BR
吲达帕 Indapamide 26807658 规格:HPLC>98%
碘帕 Iopamidol 62883005 规格:HPLC>98%,USP
碘帕 Iopamidol 62883005 规格:>98%,USP
盐洛 Loperamide HCl 34552835 规格:>98%,BR
盐洛 Loperamide HCl 34552835 规格:HPLC>99%
咯三 Ketorolac Tromethamine 74103074 规格:>98.5%,USP,BR
咯三 Ketorolac Tromethamine 74103074 规格:HPLC>98%
兰索拉唑 Lansoprazole 103577453 规格:干品含量>98%,USP32
兰索拉唑 Lansoprazole 103577453 规格:HPLC>98%
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文献和实验A method for analyzing the ubiquitination and degradation of aurora-A
has been well characterized and it was shown that it is ubiquitin proteasome pathway that leads to the elimination of cyclins. By now, many other regulatory proteins were shown to be degraded by the same pathway, among them members of the aurora kinase family, degraded
Studying the Roles of Aurora-C Kinase During Meiosis in Mouse Oocytes
We previously isolated Aurora-C (Aurkc/Aie1 ) in a screen for kinases expressed in mouse sperm and eggs. Aurora-C kinase was reported to be a chromosomal passenger protein that plays critical roles in chromosome alignment
The Ipl1/Aurora Kinase Family: Methods of Inhibition and Functional Analysis in Mammalian Cells
and the pharmaceutical industry. Indeed, two small molecule Aurora kinase inhibitors have recently been described. In this chapter, we describe several methods for investigating the function of the Aurora kinases, focusing on Aurora B. We describe the use of the small
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