Rocastine罗卡斯汀,91833-49-7

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Rocastine

CAS No. : 91833-49-7

MCE 国际站：Rocastine

产品活性：Rocastine 是一种选择性的，非镇静的 H1 拮抗剂，为抗组胺剂。

研究领域：GPCR/G Protein  |  Neuronal Signaling  |  Immunology/Inflammation

作用靶点：Histamine Receptor

In Vivo: Rocastine is effective with a 15 min pretreatment time (PD₅₀ = 0.13 mg/kg) as it is with a 1 hr pretreatment time (PD₅₀ = 0.12 mg/kg). Rocastine protects guinea pigs from collapse induced by aerosolized antigen; rocastine is approximately 36x more potent than diphenhydramine and as potent as oxatomide and terfenadine. Rocastine does not alter the EEG of cats at doses in vast excess (150x) of its antihistaminic dose nor does it potentiate yohimbine toxicity in mice.

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