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- 详细信息
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
ML414
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
790702-57-7
- 规格:
10 mM * 1 mL/1 mg/5 mg/10 mg/50 mg/100 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥550.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥250.0 |
| 规格: | 5 mg | 产品价格: | ¥500.0 |
| 规格: | 10 mg | 产品价格: | ¥800.0 |
| 规格: | 50 mg | 产品价格: | ¥2800.0 |
| 规格: | 100 mg | 产品价格: | ¥4480.0 |
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NGI-1
CAS No. : 790702-57-7
MCE 国际站:NGI-1
产品活性:NGI-1 (ML414) 是一种有效的寡糖基转移酶 (OST) 抑制剂,直接靶向和阻断 OST 催化亚基 STT3A 和 STT3B 的功能。NGI-1 是一种细胞渗透性抑制剂,可有效降低病毒感染性而不影响细胞活力。
研究领域:Anti-infection
作用靶点:Virus Protease
In Vitro: NGI-1 inhibits the glycosylation of LASV GP mediated by STT3A-OST (in STT3B- and MAGT1-TUSC3- cells) or STT3B-OST (in STT3A- cells) and impaires its proteolytic cleavage in a dose-dependent manner.
?NGI-1 blocks EGFR N-linked glycosylation in lung adenocarcinoma cells as assessed. In controls EGFR is biotinylated, consistent with its plasma membrane expression, but in NGI-1 treated cells the EGFR is predominantly found in the non-biotinylated intracellular fraction suggesting a change in cellular localization.
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