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- 详细信息
- 询价记录
- 文献和实验
- 技术资料
- 提供商:
武汉合研生物医药科技有限公司
- 服务名称:
激酶活性检测技术服务
武汉合研生物医药科技有限公司坐落于光谷生物城,是一家专注于提供新药发现阶段的技术服务,以中小微新药研发企业为服务主体的创新型公司。合研生物拥有一支训练有素的药物研发技术团队,提供的服务覆盖虚拟筛选、酶学靶点筛选、抗肿瘤药物活性评价、细胞功能学检测、药理病理学服务等各项技术,同时也提供可购买的商业化合物库。我们的技术团队在分子生物学、细胞生物学、结构生物学等领域具有丰富的经验,通过酶水平、细胞水平测定等技术平台帮助客户进行化合物筛选及化合物特性、作用机制等研究。合研生物以高效、高性价比的专业服务帮助客户更快地达到目标,帮助客户推进药物发现的进程。
我们的优势
Kinase激酶
酶学研究一直是药物研发的重要组成部分。合研生物拥有丰富的酶学筛选经验,酶学实验涵盖300多种筛选模型,包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等。根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。
| Kinase激酶 | |||
| E148 | ABL1 | ADP-Glo | 96/384 well |
| E149 | ABL1(E255K) | ADP-Glo | 96/384 well |
| E150 | ABL1(T315I) | ADP-Glo | 96/384 well |
| E151 | ABL1(Y253F) | ADP-Glo | 96/384 well |
| E152 | ACK | ADP-Glo | 96/384 well |
| E153 | AKT1 | ADP-Glo | 96/384 well |
| E154 | AKT2 | ADP-Glo | 96/384 well |
| E155 | AKT3 | ADP-Glo | 96/384 well |
| E156 | ALK2 | ADP-Glo | 96/384 well |
| E157 | ALK4 | ADP-Glo | 96/384 well |
| E158 | ALK6 | ADP-Glo | 96/384 well |
| E159 | AMAPK(A1/B1/G2) | ADP-Glo | 96/384 well |
| E160 | AMPK(A1/B1/G1) | ADP-Glo | 96/384 well |
| E161 | AMPK(A2/B1/G1) | ADP-Glo | 96/384 well |
| E162 | ASK1 | ADP-Glo | 96/384 well |
| E163 | Aurora A | ADP-Glo | 96/384 well |
| E164 | Aurora B | ADP-Glo | 96/384 well |
| E165 | AXL | ADP-Glo | 96/384 well |
| E166 | BRK | ADP-Glo | 96/384 well |
| E167 | BXM | ADP-Glo | 96/384 well |
| E168 | CAMK1γ | ADP-Glo | 96/384 well |
| E169 | CAMK2α | ADP-Glo | 96/384 well |
| E170 | CAMK2γ | ADP-Glo | 96/384 well |
| E171 | CAMKK1 | ADP-Glo | 96/384 well |
| E172 | CDC7/DBF4 | ADP-Glo | 96/384 well |
| E173 | CDK2/CyclinA2 | ADP-Glo | 96/384 well |
| E174 | CDK2/CyclinE1 | ADP-Glo | 96/384 well |
| E175 | CDK3/cyclinE1 | ADP-Glo | 96/384 well |
| E176 | CDK5/p25 | ADP-Glo | 96/384 well |
| E177 | CDK5/p35 | ADP-Glo | 96/384 well |
| E178 | CDK6/CyclinD3 | ADP-Glo | 96/384 well |
| E179 | CDK9/Cyclink | ADP-Glo | 96/384 well |
| E180 | CHK1 | ADP-Glo | 96/384 well |
| E181 | CHK2 | ADP-Glo | 96/384 well |
| E182 | CK1a1 | ADP-Glo | 96/384 well |
| E183 | CK1γ1 | ADP-Glo | 96/384 well |
| E184 | CK1ε | ADP-Glo | 96/384 well |
| E185 | CK2α1 | ADP-Glo | 96/384 well |
| E186 | c-KIT | ADP-Glo | 96/384 well |
| E187 | CLK1 | ADP-Glo | 96/384 well |
| E188 | CLK3 | ADP-Glo | 96/384 well |
| E189 | c-MER | ADP-Glo | 96/384 well |
| E190 | CSK | ADP-Glo | 96/384 well |
| E191 | DAPK1 | ADP-Glo | 96/384 well |
| E192 | DDR2 | ADP-Glo | 96/384 well |
| E193 | DNA-PK | ADP-Glo | 96/384 well |
| E194 | DYRK2 | ADP-Glo | 96/384 well |
| E195 | EGFR | ADP-Glo | 96/384 well |
| E196 | EGFR(L858R) | ADP-Glo | 96/384 well |
| E197 | EGFR(L861Q) | ADP-Glo | 96/384 well |
| E198 | EGFR(T790,L858R) | ADP-Glo | 96/384 well |
| E199 | EGFR(T790M) | ADP-Glo | 96/384 well |
| E200 | EIF2AK2 | ADP-Glo | 96/384 well |
| E201 | EPHA1 | ADP-Glo | 96/384 well |
| E202 | ERK1 | ADP-Glo | 96/384 well |
| E203 | ERK2 | ADP-Glo | 96/384 well |
| E204 | FAK | ADP-Glo | 96/384 well |
| E205 | FES | ADP-Glo | 96/384 well |
| E206 | FGFR1 | ADP-Glo | 96/384 well |
| E207 | FGFR2 | ADP-Glo | 96/384 well |
| E208 | FGFR3(K650E) | ADP-Glo | 96/384 well |
| E209 | FGFR4 | ADP-Glo | 96/384 well |
| E210 | FLT1 | ADP-Glo | 96/384 well |
| E211 | FLT3 | ADP-Glo | 96/384 well |
| E212 | FLT3(D835Y) | ADP-Glo | 96/384 well |
| E213 | FMS | ADP-Glo | 96/384 well |
| E214 | FYN A | ADP-Glo | 96/384 well |
| E215 | GRK5 | ADP-Glo | 96/384 well |
| E216 | GSK3α | ADP-Glo | 96/384 well |
| E217 | GSK3β | ADP-Glo | 96/384 well |
| E218 | HER2 | ADP-Glo | 96/384 well |
| E219 | HER4 | ADP-Glo | 96/384 well |
| E220 | HIPK1 | ADP-Glo | 96/384 well |
| E221 | HPK1 | ADP-Glo | 96/384 well |
| E222 | IGF1R | ADP-Glo | 96/384 well |
| E223 | IKKß | ADP-Glo | 96/384 well |
| E224 | IKKα | ADP-Glo | 96/384 well |
| E225 | InsR | ADP-Glo | 96/384 well |
| E226 | IRAK4 | ADP-Glo | 96/384 well |
| E227 | ITK | ADP-Glo | 96/384 well |
| E228 | JAK3 | ADP-Glo | 96/384 well |
| E229 | JNK1 | ADP-Glo | 96/384 well |
| E230 | JNK3 | ADP-Glo | 96/384 well |
| E231 | KDR | ADP-Glo | 96/384 well |
| E232 | KHS1 | ADP-Glo | 96/384 well |
| E233 | LCK | ADP-Glo | 96/384 well |
| E234 | Lipid kinase | ADP-Glo | 96/384 well |
| E235 | LRRK2 | ADP-Glo | 96/384 well |
| E236 | LYN B | ADP-Glo | 96/384 well |
| E237 | MAPKAPK2 | ADP-Glo | 96/384 well |
| E238 | MAPKAPK3 | ADP-Glo | 96/384 well |
| E239 | MAPKAPK5 | ADP-Glo | 96/384 well |
| E240 | MARK1 | ADP-Glo | 96/384 well |
| E241 | MELK | ADP-Glo | 96/384 well |
| E242 | MET | ADP-Glo | 96/384 well |
| E243 | MET(M1250T) | ADP-Glo | 96/384 well |
| E244 | MINK1 | ADP-Glo | 96/384 well |
| E245 | MLCK | ADP-Glo | 96/384 well |
| E246 | MLK1 | ADP-Glo | 96/384 well |
| E247 | MLK2 | ADP-Glo | 96/384 well |
| E248 | MRCKa | ADP-Glo | 96/384 well |
| E249 | MSK1 | ADP-Glo | 96/384 well |
| E250 | MSK2 | ADP-Glo | 96/384 well |
| E251 | MST1 | ADP-Glo | 96/384 well |
| E252 | MYO3β | ADP-Glo | 96/384 well |
| E253 | Name | ADP-Glo | 96/384 well |
| E254 | NEK2 | ADP-Glo | 96/384 well |
| E255 | NEK3 | ADP-Glo | 96/384 well |
| E256 | NIK | ADP-Glo | 96/384 well |
| E257 | NUAK2 | ADP-Glo | 96/384 well |
| E258 | p38B | ADP-Glo | 96/384 well |
| E259 | p38α | ADP-Glo | 96/384 well |
| E260 | p38γ | ADP-Glo | 96/384 well |
| E261 | P38δ | ADP-Glo | 96/384 well |
| E262 | p70S6K | ADP-Glo | 96/384 well |
| E263 | p70S6Kb | ADP-Glo | 96/384 well |
| E264 | PAK1/CDC42 | ADP-Glo | 96/384 well |
| E265 | PAK3 | ADP-Glo | 96/384 well |
| E266 | PAK4 | ADP-Glo | 96/384 well |
| E267 | PASK | ADP-Glo | 96/384 well |
| E268 | PDGFRa(D842V) | ADP-Glo | 96/384 well |
| E269 | PDGFRa(T674I) | ADP-Glo | 96/384 well |
| E270 | PDGFRα | ADP-Glo | 96/384 well |
| E271 | PDGFRβ | ADP-Glo | 96/384 well |
| E272 | PDK1 | ADP-Glo | 96/384 well |
| E273 | PI3K Lipid kinases | ADP-Glo | 96/384 well |
| E274 | PI3K-Glo | ADP-Glo | 96/384 well |
| E275 | PIM1 | ADP-Glo | 96/384 well |
| E276 | PIM2 | ADP-Glo | 96/384 well |
| E277 | PKA | ADP-Glo | 96/384 well |
| E278 | PKC | ADP-Glo | 96/384 well |
| E279 | PKCß1 | ADP-Glo | 96/384 well |
| E280 | PKCα | ADP-Glo | 96/384 well |
| E281 | PKCβII | ADP-Glo | 96/384 well |
| E282 | PKCγ | ADP-Glo | 96/384 well |
| E283 | PKCδ | ADP-Glo | 96/384 well |
| E284 | PKCε | ADP-Glo | 96/384 well |
| E285 | PKCζ | ADP-Glo | 96/384 well |
| E286 | PKCθ | ADP-Glo | 96/384 well |
| E287 | PKCι | ADP-Glo | 96/384 well |
| E288 | PKCμ | ADP-Glo | 96/384 well |
| E289 | PKD2 | ADP-Glo | 96/384 well |
| E290 | PLK1 | ADP-Glo | 96/384 well |
| E291 | PRKG1 | ADP-Glo | 96/384 well |
| E292 | PYK2 | ADP-Glo | 96/384 well |
| E293 | RET | ADP-Glo | 96/384 well |
| E294 | RET(V804L) | ADP-Glo | 96/384 well |
| E295 | RET(Y791F) | ADP-Glo | 96/384 well |
| E296 | RIPK2 | ADP-Glo | 96/384 well |
| E297 | ROCK1 | ADP-Glo | 96/384 well |
| E298 | ROCK2 | ADP-Glo | 96/384 well |
| E299 | RON | ADP-Glo | 96/384 well |
| E300 | RSK1 | ADP-Glo | 96/384 well |
| E301 | SGK1 | ADP-Glo | 96/384 well |
| E302 | SIK | ADP-Glo | 96/384 well |
| E303 | SLK | ADP-Glo | 96/384 well |
| E304 | SRC | ADP-Glo | 96/384 well |
| E305 | STK33 | ADP-Glo | 96/384 well |
| E306 | SYK | ADP-Glo | 96/384 well |
| E307 | TAK1-TAB1 | ADP-Glo | 96/384 well |
| E308 | TAOK1 | ADP-Glo | 96/384 well |
| E309 | TBK1 | ADP-Glo | 96/384 well |
| E310 | TGFbR1 | ADP-Glo | 96/384 well |
| E311 | TGFβR2 | ADP-Glo | 96/384 well |
| E312 | TNIK | ADP-Glo | 96/384 well |
| E313 | TOPK | ADP-Glo | 96/384 well |
| E314 | TRKA | ADP-Glo | 96/384 well |
| E315 | TRKB | ADP-Glo | 96/384 well |
| E316 | ULK1 | ADP-Glo | 96/384 well |
| E317 | VRK2 | ADP-Glo | 96/384 well |
| E318 | WNK1 | ADP-Glo | 96/384 well |
| E319 | ZAK | ADP-Glo | 96/384 well |
| E320 | ZAP70 | ADP-Glo | 96/384 well |
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文献和实验Western Blot 实验 通过SDS-PAGE胶将不同的分子量的蛋白分离开,将目标蛋白转移到PVDF膜上,再利用抗原抗体的特异性结合,用特异性的一抗结合目标蛋白,用HRP标记的二抗结合一抗,再加以ECL发光液显色,检测目的蛋白在不同处理的样本中表达量的高低变化 服务优势及实验服务流程: 1、利用高性能试剂配合高通量全自动western blot机,提供超高灵敏性的western blot实验服务。超高灵敏度最低至15飞克抗原。 2、一抗的寄送需要泡沫盒加冰袋低温即送
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yan0495 R&D公司的recombinant human EGF Receptor来源于DNA编码的人类EGFR的胞外区,而酪氨酸激酶活性区在胞内,我现在需要做酪氨酸激酶抑制剂的筛选,不知道能不能用这个蛋白?筛选原理: 以多聚酪氨酸多肽为底物,用EGFR催化酪氨酸的磷酸化,用酶标记的单克隆抗体检测酪氨酸磷酸化程度,以OPD做为辣根过氧化物酶底物显色,从而筛选EGFR抑制剂。附上EGFR说明书和图。 请各位指点啊! yan








