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酶学靶点抑制剂筛选---激酶

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  • 询价
  • 靶点抑制剂筛选
  • 武汉
  • 2026年01月19日
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    武汉合研生物医药科技有限公司
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    • 提供商：

      合研生物

    • 服务名称：

      激酶抑制剂活性筛选

     公司介绍

            武汉合研生物医药科技有限公司坐落于光谷生物城，是一家专注于提供新药发现阶段的技术服务，以中小微新药研发企业为服务主体的创新型公司。合研生物拥有一支训练有素的药物研发技术团队，提供的服务覆盖虚拟筛选、酶学靶点筛选、抗肿瘤药物活性评价、细胞功能学检测、药理病理学服务等各项技术。我们的技术团队在分子生物学、细胞生物学、结构生物学等领域具有丰富的经验，通过酶水平、细胞水平测定等技术平台帮助客户进行化合物筛选及化合物特性、作用机制等研究。合研生物以高效、高性价比的专业服务帮助客户更快地达到目标，帮助客户推进药物发现的进程。

    我们的服务

    Kinase激酶
            酶学研究一直是药物研发的重要组成部分。合研生物拥有丰富的酶学筛选经验，酶学实验涵盖300多种筛选模型，包括了常见的组蛋白去乙酰酶类，组蛋白去甲基化酶，酪氨酸激酶，丝氨酸激酶，甲基化转移酶，磷酸二酯酶，DNA修复酶，热休克蛋白，免疫相关蛋白等。根据样本量的大小提供灵活的项目实施安排计划，可提供96孔和384孔两种板型的筛选模式，加速您的药物研发进程。
    Kinase激酶 　 　 　
    E148 ABL1 ADP-Glo 96/384 well
    E149 ABL1(E255K) ADP-Glo 96/384 well
    E150 ABL1(T315I) ADP-Glo 96/384 well
    E151 ABL1(Y253F) ADP-Glo 96/384 well
    E152 ACK ADP-Glo 96/384 well
    E153 AKT1 ADP-Glo 96/384 well
    E154 AKT2 ADP-Glo 96/384 well
    E155 AKT3 ADP-Glo 96/384 well
    E156 ALK2 ADP-Glo 96/384 well
    E157 ALK4 ADP-Glo 96/384 well
    E158 ALK6 ADP-Glo 96/384 well
    E159 AMAPK(A1/B1/G2) ADP-Glo 96/384 well
    E160 AMPK(A1/B1/G1) ADP-Glo 96/384 well
    E161 AMPK(A2/B1/G1) ADP-Glo 96/384 well
    E162 ASK1 ADP-Glo 96/384 well
    E163 Aurora A ADP-Glo 96/384 well
    E164 Aurora B ADP-Glo 96/384 well
    E165 AXL ADP-Glo 96/384 well
    E166 BRK ADP-Glo 96/384 well
    E167 BXM ADP-Glo 96/384 well
    E168 CAMK1γ ADP-Glo 96/384 well
    E169 CAMK2α ADP-Glo 96/384 well
    E170 CAMK2γ ADP-Glo 96/384 well
    E171 CAMKK1 ADP-Glo 96/384 well
    E172 CDC7/DBF4 ADP-Glo 96/384 well
    E173 CDK2/CyclinA2 ADP-Glo 96/384 well
    E174 CDK2/CyclinE1 ADP-Glo 96/384 well
    E175 CDK3/cyclinE1 ADP-Glo 96/384 well
    E176 CDK5/p25 ADP-Glo 96/384 well
    E177 CDK5/p35 ADP-Glo 96/384 well
    E178 CDK6/CyclinD3 ADP-Glo 96/384 well
    E179 CDK9/Cyclink ADP-Glo 96/384 well
    E180 CHK1 ADP-Glo 96/384 well
    E181 CHK2 ADP-Glo 96/384 well
    E182 CK1a1 ADP-Glo 96/384 well
    E183 CK1γ1 ADP-Glo 96/384 well
    E184 CK1ε ADP-Glo 96/384 well
    E185 CK2α1 ADP-Glo 96/384 well
    E186 c-KIT ADP-Glo 96/384 well
    E187 CLK1 ADP-Glo 96/384 well
    E188 CLK3 ADP-Glo 96/384 well
    E189 c-MER ADP-Glo 96/384 well
    E190 CSK ADP-Glo 96/384 well
    E191 DAPK1 ADP-Glo 96/384 well
    E192 DDR2 ADP-Glo 96/384 well
    E193 DNA-PK ADP-Glo 96/384 well
    E194 DYRK2 ADP-Glo 96/384 well
    E195 EGFR ADP-Glo 96/384 well
    E196 EGFR(L858R) ADP-Glo 96/384 well
    E197 EGFR(L861Q) ADP-Glo 96/384 well
    E198 EGFR(T790,L858R) ADP-Glo 96/384 well
    E199 EGFR(T790M) ADP-Glo 96/384 well
    E200 EIF2AK2 ADP-Glo 96/384 well
    E201 EPHA1 ADP-Glo 96/384 well
    E202 ERK1 ADP-Glo 96/384 well
    E203 ERK2 ADP-Glo 96/384 well
    E204 FAK ADP-Glo 96/384 well
    E205 FES ADP-Glo 96/384 well
    E206 FGFR1 ADP-Glo 96/384 well
    E207 FGFR2 ADP-Glo 96/384 well
    E208 FGFR3(K650E) ADP-Glo 96/384 well
    E209 FGFR4 ADP-Glo 96/384 well
    E210 FLT1 ADP-Glo 96/384 well
    E211 FLT3 ADP-Glo 96/384 well
    E212 FLT3(D835Y) ADP-Glo 96/384 well
    E213 FMS ADP-Glo 96/384 well
    E214 FYN A ADP-Glo 96/384 well
    E215 GRK5 ADP-Glo 96/384 well
    E216 GSK3α ADP-Glo 96/384 well
    E217 GSK3β ADP-Glo 96/384 well
    E218 HER2 ADP-Glo 96/384 well
    E219 HER4 ADP-Glo 96/384 well
    E220 HIPK1 ADP-Glo 96/384 well
    E221 HPK1 ADP-Glo 96/384 well
    E222 IGF1R ADP-Glo 96/384 well
    E223 IKKß ADP-Glo 96/384 well
    E224 IKKα ADP-Glo 96/384 well
    E225 InsR ADP-Glo 96/384 well
    E226 IRAK4 ADP-Glo 96/384 well
    E227 ITK ADP-Glo 96/384 well
    E228 JAK3 ADP-Glo 96/384 well
    E229 JNK1 ADP-Glo 96/384 well
    E230 JNK3 ADP-Glo 96/384 well
    E231 KDR ADP-Glo 96/384 well
    E232 KHS1 ADP-Glo 96/384 well
    E233 LCK ADP-Glo 96/384 well
    E234 Lipid kinase ADP-Glo 96/384 well
    E235 LRRK2 ADP-Glo 96/384 well
    E236 LYN B ADP-Glo 96/384 well
    E237 MAPKAPK2 ADP-Glo 96/384 well
    E238 MAPKAPK3 ADP-Glo 96/384 well
    E239 MAPKAPK5 ADP-Glo 96/384 well
    E240 MARK1 ADP-Glo 96/384 well
    E241 MELK ADP-Glo 96/384 well
    E242 MET ADP-Glo 96/384 well
    E243 MET(M1250T) ADP-Glo 96/384 well
    E244 MINK1 ADP-Glo 96/384 well
    E245 MLCK ADP-Glo 96/384 well
    E246 MLK1 ADP-Glo 96/384 well
    E247 MLK2 ADP-Glo 96/384 well
    E248 MRCKa ADP-Glo 96/384 well
    E249 MSK1 ADP-Glo 96/384 well
    E250 MSK2 ADP-Glo 96/384 well
    E251 MST1 ADP-Glo 96/384 well
    E252 MYO3β ADP-Glo 96/384 well
    E253 Name ADP-Glo 96/384 well
    E254 NEK2 ADP-Glo 96/384 well
    E255 NEK3 ADP-Glo 96/384 well
    E256 NIK ADP-Glo 96/384 well
    E257 NUAK2 ADP-Glo 96/384 well
    E258 p38B ADP-Glo 96/384 well
    E259 p38α ADP-Glo 96/384 well
    E260 p38γ ADP-Glo 96/384 well
    E261 P38δ ADP-Glo 96/384 well
    E262 p70S6K ADP-Glo 96/384 well
    E263 p70S6Kb ADP-Glo 96/384 well
    E264 PAK1/CDC42 ADP-Glo 96/384 well
    E265 PAK3 ADP-Glo 96/384 well
    E266 PAK4 ADP-Glo 96/384 well
    E267 PASK ADP-Glo 96/384 well
    E268 PDGFRa(D842V) ADP-Glo 96/384 well
    E269 PDGFRa(T674I) ADP-Glo 96/384 well
    E270 PDGFRα ADP-Glo 96/384 well
    E271 PDGFRβ ADP-Glo 96/384 well
    E272 PDK1 ADP-Glo 96/384 well
    E273 PI3K Lipid kinases ADP-Glo 96/384 well
    E274 PI3K-Glo ADP-Glo 96/384 well
    E275 PIM1 ADP-Glo 96/384 well
    E276 PIM2 ADP-Glo 96/384 well
    E277 PKA ADP-Glo 96/384 well
    E278 PKC ADP-Glo 96/384 well
    E279 PKCß1 ADP-Glo 96/384 well
    E280 PKCα ADP-Glo 96/384 well
    E281 PKCβII ADP-Glo 96/384 well
    E282 PKCγ ADP-Glo 96/384 well
    E283 PKCδ ADP-Glo 96/384 well
    E284 PKCε ADP-Glo 96/384 well
    E285 PKCζ ADP-Glo 96/384 well
    E286 PKCθ ADP-Glo 96/384 well
    E287 PKCι ADP-Glo 96/384 well
    E288 PKCμ ADP-Glo 96/384 well
    E289 PKD2 ADP-Glo 96/384 well
    E290 PLK1 ADP-Glo 96/384 well
    E291 PRKG1 ADP-Glo 96/384 well
    E292 PYK2 ADP-Glo 96/384 well
    E293 RET ADP-Glo 96/384 well
    E294 RET(V804L) ADP-Glo 96/384 well
    E295 RET(Y791F) ADP-Glo 96/384 well
    E296 RIPK2 ADP-Glo 96/384 well
    E297 ROCK1 ADP-Glo 96/384 well
    E298 ROCK2 ADP-Glo 96/384 well
    E299 RON ADP-Glo 96/384 well
    E300 RSK1 ADP-Glo 96/384 well
    E301 SGK1 ADP-Glo 96/384 well
    E302 SIK ADP-Glo 96/384 well
    E303 SLK ADP-Glo 96/384 well
    E304 SRC ADP-Glo 96/384 well
    E305 STK33 ADP-Glo 96/384 well
    E306 SYK ADP-Glo 96/384 well
    E307 TAK1-TAB1 ADP-Glo 96/384 well
    E308 TAOK1 ADP-Glo 96/384 well
    E309 TBK1 ADP-Glo 96/384 well
    E310 TGFbR1 ADP-Glo 96/384 well
    E311 TGFβR2 ADP-Glo 96/384 well
    E312 TNIK ADP-Glo 96/384 well
    E313 TOPK ADP-Glo 96/384 well
    E314 TRKA ADP-Glo 96/384 well
    E315 TRKB ADP-Glo 96/384 well
    E316 ULK1 ADP-Glo 96/384 well
    E317 VRK2 ADP-Glo 96/384 well
    E318 WNK1 ADP-Glo 96/384 well
    E319 ZAK ADP-Glo 96/384 well
    E320 ZAP70 ADP-Glo 96/384 well


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