CGP 7930

概述

• 产品名称
  CGP 7930
• 描述
  Positive GABA_B receptor allosteric modulator
• 生物学描述
  Positive GABA_B receptor allosteric modulator (EC₅₀ values are 5.37 and 4.60 μM, respectively). Increases receptor agonist affinity and signal transduction efficacy. Also shown to potentiate receptor response to baclofen (ab120325).
• 纯度
  > 98%

性能

• 化学名称
  3,5-Bis(1,1-dimethylethyl)-4-hydroxy-β,β-dimethylbenzenepropanol
• 分子量
  292.46
• 化学结构
  
• 分子式
  C₁₉H₃₂O₂
• CAS编号
  57717-80-3
• PubChem识别号
  5024764
• 存放说明
  Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months.
• 溶解度概述
  Soluble in DMSO to 100 mM and in ethanol to 100 mM
• 处理

  Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

  Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

• SMILES
  CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CC(C)(C)CO
• 来源

  Synthetic