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- 详细信息
- 技术资料
- 保存条件:
-20°C
- 保质期:
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -3052℃ for several months.
- 英文名:
Ruxolitinib (INCB-18424) phosphate
- 库存:
详询
- 供应商:
详询
- CAS号:
1092939-17-7
- 规格:
5mg/10mg/25mg/50mg/1ml/10mM
| 规格: | 5mg | 产品价格: | ¥672.0 |
|---|---|---|---|
| 规格: | 10mg | 产品价格: | ¥1167.0 |
| 规格: | 25mg | 产品价格: | ¥1891.0 |
| 规格: | 50mg | 产品价格: | ¥2863.0 |
| 规格: | 1ml/10mM | 产品价格: | ¥669.0 |
ID:T3043
PURITY:1
Formula:C17H21N6O4P
MolWt:404.36
Appearance:白色粉末
Solubility:G4100 mM in DMSO
Bioactivity:Ruxolitinib phosphate(INCB018424 phosphate) is the first potent, selective, JAK1/2 inhibitor to enter the clinic with IC50 of 3.3 nM/2.8 nM, >130-fold selectivity for JAK1/2 versus JAK3.
Status:FDA
Pathways:JAK/STAT Signaling
Target:JAK inhibitor
Receptor:JAK1/2
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