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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
-20°C
- 保质期:
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -1930℃ for several months.
- 英文名:
RKI-1447
- 库存:
详询
- 供应商:
详询
- CAS号:
1342278-01-6
- 规格:
5mg/10mg/50mg/100mg/1ml/10mM
| 规格: | 5mg | 产品价格: | ¥795.0 |
|---|---|---|---|
| 规格: | 10mg | 产品价格: | ¥1125.0 |
| 规格: | 50mg | 产品价格: | ¥3232.0 |
| 规格: | 100mg | 产品价格: | ¥5483.0 |
| 规格: | 1ml/10mM | 产品价格: | ¥791.0 |
ID:T1898
PURITY:0.98
Formula:C16H14N4O2S
MolWt:326.37
Appearance:类白色粉末
Solubility:G410 mM in DMSO
Bioactivity:RKI-1447 is a potent inhibitor of ROCK1 and ROCK2, with IC50 of 14.5 nM and 6.2 nM, respectively, has anti-invasive and antitumor activities.
Status:
Pathways:Cell Cycle/Checkpoint
Target:ROCK inhibitor
Receptor:ROCK1/2
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文献和实验A Neurovascular BloodBrain Barrier In Vitro Model
Clin Invest 113:1447–1455, 2004), or formation of oxidative stress (Yemisci et al., Nat Med 15:1031–1037, 2009). Hence, this interdependent assembly of cells is referred to as the neurovascular unit (NVU) (Zlokovic, Nat Med 16:1370–1371, 2010; Zlokovic
0.3325 0.3318 0.3306 0.3290 0.3273 0.3253 0.3232 0.3211 3 0.2260 0.2347 0.2412 0.2460 0.2495 0.2521 0.2540 0.2553 0.2561 0.2565 4 0.1429 0.1586 0.1707 0.1802 0.1878 0.1939 0.1988 0.2027 0.2059 0.2085 5 0.0695 0.0922 0.1099 0.1240 0.1353 0.1447 0.1524
) 65122268-1447,E-mail: cmajy@public.sti.ac.cn(10)临床检验杂志(LINCHUANG JIANYAN ZAZHI,Chinese journal of clinical laboratory science)编辑部地址: 南京市中央路42号,邮编:210008电话:(025)7714280,E-mail: jcls@publicl.ptt.js.cn(11)上海医学检验杂志(SHANGHAI YIXUE JIANYAN ZAZHI,Shanghai Journal
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