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- 详细信息
- 技术资料
- 保存条件:
-20°C
- 保质期:
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -1823℃ for several months.
- 英文名:
Regorafenib (BAY 73-4506)
- 库存:
详询
- 供应商:
详询
- CAS号:
755037-03-7
- 规格:
5mg/10mg/25mg/50mg/100mg/1ml/10mM
| 规格: | 5mg | 产品价格: | ¥418.0 |
|---|---|---|---|
| 规格: | 10mg | 产品价格: | ¥757.0 |
| 规格: | 25mg | 产品价格: | ¥1088.0 |
| 规格: | 50mg | 产品价格: | ¥1891.0 |
| 规格: | 100mg | 产品价格: | ¥3403.0 |
| 规格: | 1ml/10mM | 产品价格: | ¥368.0 |
ID:T1792
PURITY:0.98
Formula:C21H15ClF4N4O3
MolWt:482.82
Appearance:白色粉末
Solubility:G4DMSO > 100mM
Bioactivity:Regorafenib (BAY 73-4506) is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM in cell-free assays, respectively.
Status:
Pathways:Tyrosine Kinase/Adaptors; MAPK Signaling
Target:VEGFR inhibitor; PDGFR inhibitor; FGFR inhibitor; Raf inhibitor
Receptor:VEGFR1/2/3;PDGFRβ;FGFR; Raf-1/B-Raf
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