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- 详细信息
- 文献和实验
- 技术资料
- 库存:
详询
- 英文名:
TAK-593
- CAS号:
1005780-62-0
- 保质期:
Powder:2-8℃,2 years;Insolvent(母液):-20℃,6 months;-80℃,1 year
- 供应商:
北京索莱宝科技有限公司
- 保存条件:
Powder:2-8℃,2 years;Insolvent(母液):-20℃,6 months;-80℃,1 year
- 规格:
1mg/5mg/10mg/25mg/100mg
| 规格: | 1mg | 产品价格: | ¥482.0 |
|---|---|---|---|
| 规格: | 5mg | 产品价格: | ¥1052.0 |
| 规格: | 10mg | 产品价格: | ¥1814.0 |
| 规格: | 25mg | 产品价格: | ¥3714.0 |
| 规格: | 100mg | 产品价格: | ¥5440.0 |
靶点 PDGFR;VEGFR
通路 Angiogenesis; Protein Tyrosine Kinase/RTK
背景说明 TAK-593是有效的 VEGFR2 和 PDGFR 抑制剂。




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文献和实验[1]. Miyamoto N, et al. Discovery of N-[5-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)-2-methylphenyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide (TAK-593), a highly potent VEGFR2 kinase inhibitor. Bioorg Med Chem. 2013 Apr 15;21(8):2333-2345.
[2]. Awazu Y, et al. Anti-angiogenic and anti-tumor effects of TAK-593, a potent and selective inhibitor of vascular endothelial growth factor and platelet-derived growth factor receptor tyrosine kinase. Cancer Sci. 2013 Apr;104(4):486-94.
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V294.PART II,Chapter 4 细胞迁移实验之Dunn趋化迁移培养皿法及时序显微镜分析法
, the DCC has been used to study neurite outgrowth(12). We have previously used the DCC to elucidate the role of Rho family proteinsin the chemotactic response of BAC1.2F5 macrophages to CSF-1 (13). Wedescribe the use of this chamber to study the response
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