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- 详细信息
- 技术资料
- 保存条件:
零下80~20°C
- 保质期:
Powder: -20°C for 3 years In solvent: -80°C for 2 years
- 英文名:
FNDR-20123
- 库存:
10
- 供应商:
TargetMol
- 规格:
25 mg/100 mg/50 mg
| 规格: | 25 mg | 产品价格: | ¥11400.0 |
|---|---|---|---|
| 规格: | 100 mg | 产品价格: | ¥23700.0 |
| 规格: | 50 mg | 产品价格: | ¥14900.0 |
Product Introduction
Bioactivity
英文名:FNDR-20123
描述:FNDR-20123 is the first safe and effective anti-malarial HDAC inhibitor, acting on both Plasmodium falciparum HDAC (IC50: 31 nM) and human HDAC (IC50: 3 nM). FNDR-20123 inhibited HDAC1 (IC50: 25 nM), HDAC2 (IC50: 29 nM), HDAC3 (IC50: 2 nM), HDAC6 (IC50: 11 nM), HDAC8 (IC50: 282 nM) and, at nanomolar concentrations, HDAC3 (IC50: 2 nM). The inhibitor of HDAC subtype III was also observed at nanomolar concentrations.

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FNDR-20123
¥11400 - 23700







