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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
零下80~20°C
- 保质期:
Powder: -20°C for 3 years In solvent: -80°C for 2 years
- 英文名:
NFATc1-IN-1
- 库存:
10
- 供应商:
TargetMol
- CAS号:
1912422-56-0
- 规格:
25 mg/10 mg/5 mg/50 mg/100 mg/500 mg/1 mg
| 规格: | 25 mg | 产品价格: | ¥1660.0 |
|---|---|---|---|
| 规格: | 10 mg | 产品价格: | ¥821.0 |
| 规格: | 5 mg | 产品价格: | ¥467.0 |
| 规格: | 50 mg | 产品价格: | ¥2490.0 |
| 规格: | 100 mg | 产品价格: | ¥3730.0 |
| 规格: | 500 mg | 产品价格: | ¥7880.0 |
| 规格: | 1 mg | 产品价格: | ¥213.0 |
Product Introduction
Bioactivity
英文名:NFATc1-IN-1
描述:NFATc1-IN-1 (also known as compound A04) is a highly effective inhibitor of osteoclast formation induced by RANKL, with an IC50 of 1.57 μM. It exerts its anti-osteoclastogenic effects by attenuating the RANKL-induced nuclear translocation of NFATc1. Due to its remarkable properties, NFATc1-IN-1 holds significant potential for advancing research related to osteoclastic diseases [1].

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文献和实验-Abl,Bax,CrkII,TAK1,ASK1,MAPKKKs,HPK1,GCK,MEKK1,MEKK4,MLK2,MLK3,DLK,TpI-2,TAO1,TAO2,PI3Kγ,c-Jun,SOS,Ras,TRAF2,Daxx,POSH,MLKs,MKPs,NFATc1,Gα12,Gβγ,JIP1,JIP2,JIP3,ATF-2,Elk-1,Smad4,p53,NFAT4,Stat3,Rac,Cdc42,Rho,HSF1,Gα13,14-3-3等
14. MKK: MAP2K1, MAP2K2, MAP2K3, MAP2K4, MAP2K5, MAP2K6, MAP2K7. MKKK: ARAF1, BRAF, DLK1, MAP3K1, MAP3K2, MAP3K3, MAP3K4, MAP3K5, MAP3K7, MAP3K11, MAP3K14, MAP4K1, MAP4K3, MOS, MST1, PAK1, PAK3, RAF1. NFAT Family Members: NFATC1, NFATC2, NFATC3
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