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- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
2427608-43-1
- 规格:
10 mM * 1 mL///1 mg
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JAK1-IN-11
CAS No. : 2427608-43-1
MCE 国际站:JAK1-IN-11
产品活性:JAK1-IN-11 (compound 11) 是一种有效的 JAK 抑制剂,IC50 为 0.02 nM (JAK1) 和 0.44 nM (JAK2)。JAK1-IN-11 对 JAK1 的选择性高于 JAK2。
研究领域:Epigenetics | Protein Tyrosine Kinase/RTK | JAK/STAT Signaling | Stem Cell/Wnt
作用靶点:JAK
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文献和实验growth factors initiates receptor dimerization and subsequent events to activate these intraCell ular pathways. AKT is activated downstream of PI3K and has multiple targets. AKT and the cellular energy sensors LKB1 (STK11) and AMP-activated protein
2R5C, PPP2R5D, PPP2R5E, PTEN, PRKCA, PRKCB1, PRKCZ, TCL1A, TCL1B. JAK and STAT Proteins: JAK1, JAK2, JAK3, STAT1, STAT2, STAT3, STAT4, STAT5A, STAT5B, STAT6, TYK2. MAPK: MAPK1, MAPK3, MAPK6, MAPK7, MAPK8, MAPK9, MAPK10, MAPK11, MAPK12, MAPK13, MAPK
5(extracellular signal-regulated kinase) JNK(c-Jun N-terminal kinase), P38, etc. (11)MOS/Raf protein kinase 2.蛋白酪氨酸激酶 (1) Growth factor receptors
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