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- 库存:
99
- 英文名:
Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit
- 供应商:
北京云肽生物科技有限公司
Cayman 10011671 可溶性环氧化物水解酶抑制剂筛选试剂盒-96次分析,Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit
Cayman ( 美国 )
Cayman Chemical向全球科学工作者提供多研究领域的生化、免疫试剂和分析试剂盒,其产品被广泛应用于肿瘤、氧化氮、神经学、凋亡、氧化性损伤、内分泌学等不同研究领域。
Cayman Chemical可提供用于检测的特色试剂盒,如:类花生酸类物质、游离的生物标志、环核苷、激素及氧化氮等;也提供多种高质量试剂,包括:类花生酸类物 质、氧化氮试剂及许多相关脂质、脂肪酸、酶和抗体。
Cayman Chemical在位于密西根安娜堡(Ann Arbor, Michigan)66,000平方英尺的工厂生产并制作近6000多种不同的化合物、抗体及分析试剂盒。
我们北京云肽生物科技有限公司作为Cayman公司的经销商为客户提供,正规进口,保证原装正品,货期稳定,折扣好的服务标准
Cayman 10011671 Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit可溶性环氧化物水解酶抑制剂筛选试剂盒-96次分析,产品简介:
产品品牌:Cayman
产品名称:可溶性环氧化物水解酶抑制剂筛选试剂盒-96次分析
英文名称:Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit
产品货号:10011671
产品规格:96 wells
Cayman 10011671 Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit可溶性环氧化物水解酶抑制剂筛选试剂盒-96次分析,产品说明:
可溶性环氧化物水解酶(sEH)催化外源和内源环氧化物水解为邻二醇。sEH的内源性底物包括具有血管舒张和抗炎活性的环氧二十碳三烯酸(EET)。因此,sEH的小分子抑制剂有望成为治疗高血压和血管炎症的药物。Cayman基于荧光的sEH抑制剂筛选分析试剂盒为筛选环氧化物水解酶抑制剂提供了一种方便的方法。该分析利用(3-苯基-环氧yi烷基)-乙酸qing基-(6-甲氧基-萘-2-基)-甲酯(PHOME)作为底物。
通过环氧化物水解酶水解PHOME产生高荧光6-甲氧基-2-萘甲醛,可使用330 nm的激发波长和465 nm的发射波长对其进行分析。每个试剂盒包含缓冲液、底物和足够的人类重组sEH,可用于100次试验。
可溶性环氧化物水解酶(sEH)是一种能代谢环氧脂肪酸的酶,它在哺乳动物中广泛存在,能将内源性环氧二十碳三烯酸(EETs)转化为二羟基二十碳三烯酸(DHETs).内源性EETs是由花生四烯酸(AA)经细胞色素P450氧化而来,它是生物体内重要的信号分子,具有调节离子转运和基因表达、血管扩张、抗炎等作用.在动物体内,有很多种途径可以降解EETs,其中sEH将EETs代谢为DHETs是最主要的代谢途径,使EETs的浓度降低,生理活性下降,从而使体内的血压升高,并进一步影响肾脏,心脏等功能.研究表明,抑制sEH的活性可治疗多种心血管疾病及炎症.
警告:本产品不供人类或兽医使用。
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Cayman 10008187 Dimethylcurcumin 1 mg
Cayman 10008187 Dimethylcurcumin 10 mg
Cayman 10008187 Dimethylcurcumin 25 mg
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Cayman 10011619 Terbinafine (hydrochloride) 250 mg
Cayman 10011619 Terbinafine (hydrochloride) 500 mg
Cayman 10011620 Raloxifene (hydrochloride) 100 mg
Cayman 10011620 Raloxifene (hydrochloride) 250 mg
Cayman 10011620 Raloxifene (hydrochloride) 50 mg
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Cayman10011671可溶性环氧化物水解酶抑制剂筛选试剂盒-96次分析,Soluble Epoxide Hydrolase Inhibitor Screening Assay Kit
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