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- 保存条件:
-20°C, protect from light
- 英文名:
PF-00299804-d<sub>10</sub> dihydrochloride; PF-299804-d<sub>10</sub> dihydrochloride
- 库存:
货期:14天
- 供应商:
MedChemExpress LLC
- 规格:
1 mg///5 mg
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Dacomitinib-d10 dihydrochloride
MCE 国际站:Dacomitinib-d10 dihydrochloride
产品活性:Dacomitinib-d10 (dihydrochloride) 是 Dacomitinib dihydrochloride 的氘代物。Dacomitinib (PF-00299804) dihydrochloride 是一种特异,不可逆的 ERBB 家族抑制剂,作用于 EGFR,ERBB2 和 ERBB4 的 IC50 分别为 6 nM,45.7 nM 和 73.7 nM
研究领域:Others | JAK/STAT Signaling | Protein Tyrosine Kinase/RTK | Apoptosis
作用靶点:Isotope-Labeled Compounds | EGFR | Apoptosis
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
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Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Dye Reagents | PROTAC | Isotope-Labeled Compounds
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文献和实验疟原虫 Malaria Parasites(Plasmodium)
can be used:Quinine dihydrochloride 20 mg salt/kg base given I.V. in 5% w/v dextrose or normal saline as a once-only 4 hour infusion followed, 4 hours later, by quinine dihydrochloride 10 mg salt/kg base 4-hour infusions 8 hourly.Where a syringe pump
” 两把效果一样但又能互补的 “剪刀”,作为 “厨师” 的我们,只要能达到我们的目标,选择任一 “剪刀” 都可。1.5 利用 CRISPR/Cas 系统在基因组编辑方式上的技术创新1.5.1 植物基因组单碱基编辑系统创新和应用单碱基突变可引起作物许多农艺性状的改变,因此,实施单碱基编辑对作物遗传改良具有十分重要的意义。2016 年 5 月,《Nature》报道了 KOMOR 等将大鼠胞嘧啶脱氨酶 (APOBEC1,一种碱基修饰酶能改变 DNA 序列)、Cas9 变体 (D10A) 和尿嘧啶糖
ml warm D10 onto plate and place in incubator. 36-48 hours after transfection, harvest viral supernatant and spin at 2000 rpm, 7 min at 4� in a 50ml tube. Filter viral SN through .45 um filter. Add 35ml of filtered
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