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- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
E7080-d<sub>4</sub>
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- 规格:
500 μg/1 mg
| 规格: | 500 μg | 产品价格: | ¥3600.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥5400.0 |
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Lenvatinib-d4
CAS No. : 2264050-65-7
MCE 国际站:Lenvatinib-d4
产品活性:Lenvatinib-d4 是 Lenvatinib 的氘代物。Lenvatinib (E7080) 一种具有口服活性的,多靶点酪氨酸激酶抑制剂,抑制血管内皮生长因子受体 (VEGFR1-3),成纤维细胞生长因子受体 (FGFR1-4),血小板衍生生长因子受体 (PDGFR),干细胞因子受体 (KIT),转染期间重排 (RET),显示有效抗癌的活性。
研究领域:Protein Tyrosine Kinase/RTK
作用靶点:VEGFR | FGFR | PDGFR | c-Kit | RET
In Vitro: Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
相关产品:Sorafenib | Lenvatinib | Pexidartinib | Sunitinib | Regorafenib | Nintedanib | Bevacizumab | Imatinib | Semaxinib | Cabozantinib | Ponatinib | Erdafitinib | Infigratinib | Axitinib | Midostaurin | Pemigatinib | Chloramphenicol | Pazopanib | Futibatinib | Fexagratinib | PD173074 | Pralsetinib | Selpercatinib | Heparan Sulfate | Formononetin | Crenolanib | 5Z-7-Oxozeaenol | Linifanib
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Characterization of Dopamine Receptors
of the radioligand's molar concentration is also included. Keywords: Receptor binding; dopamine; D1; D2; D3; D4; D5; radioligand binding GO TO THE FULL PROTOCOL:
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