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- 文献和实验
- 技术资料
- 保存条件:
Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
- 英文名:
RM-023
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- 规格:
10 mM * 1 mL/1 mg/5 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥4949.0 |
|---|---|---|---|
| 规格: | 1 mg | 产品价格: | ¥1850.0 |
| 规格: | 5 mg | 产品价格: | ¥4500.0 |
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RMC-0331
CAS No. : 2488788-52-7
MCE 国际站:RMC-0331
产品活性:RMC-0331 (RM-023) 是一种高效、选择性和口服生物利用度 SOS1 抑制剂。RMC-0331 是一种体内工具化合物,通过破坏 RAS-SOS1 相互作用阻断 RAS 激活。
研究领域:Protein Tyrosine Kinase/RTK | GPCR/G Protein
In Vitro: RMC-0331 has an IC50 of 71 nM measuring by the rate of GDP/GTP exchange in vitro.
In Vivo: RMC-0331 (100-250 mg/kg; p.o.; qd; immunocompetent mice) shows single agent anti-tumor activity in SHP2-mutant models.
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文献和实验大多数白细胞分化抗原在生物进化中具有保守性,这是不同种属动物执行相同或相似生物学功能的需要。小鼠是免疫学研究中最常用的实验动物,而且对某些人白细胞分化抗原的结构和功能的了解首先是从小鼠或小鼠源性的细胞实验模型得知的。目前已有小鼠CD编号及鉴定出的相应mAb(见附表1),但在应用小鼠CD分子或mAb时应注意以下三方面问题。(一) 某些人CD分子尚未在小鼠中确定迄今为止,约有30多个人CD分子尚未在小鼠中鉴定出,包括:CD15、CD17、CD39、CD42、CD46、CD52、CD57、CD
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Generation of Spatio‐Temporally Controlled Targeted Somatic Mutations in the Mouse
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