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- 详细信息
- 文献和实验
- 技术资料
- 保存条件:
4°C, sealed storage, away from moisture
- 英文名:
BTRX-246040 tartrate
- 库存:
货期:1-2天
- 供应商:
MedChemExpress LLC
- CAS号:
1307245-87-9
- 规格:
10 mM * 1 mL/5 mg/10 mg/25 mg
| 规格: | 10 mM * 1 mL | 产品价格: | ¥2777.0 |
|---|---|---|---|
| 规格: | 5 mg | 产品价格: | ¥2000.0 |
| 规格: | 10 mg | 产品价格: | ¥3488.0 |
| 规格: | 25 mg | 产品价格: | ¥5960.0 |
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LY2940094 tartrate
CAS No. : 1307245-87-9
MCE 国际站:LY2940094 tartrate
产品活性:LY2940094 (BTRX-246040) tartrate 是一种高效、可透过大脑的、选择性、口服的 NOP 受体拮抗剂,具有高亲和力 (Ki=0.105 nM) 和拮抗作用 (Kb=0.166 nM)。LY2940094 tartrate 可减少动物模型中的乙醇自我给药和寻求乙醇。
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:Opioid Receptor
In Vivo: LY2940094 (3, 10, or 30 mg/kg; orally daily for 4 days) dose-dependently reduces homecage ethanol self-administration in Indiana Alcohol-Preferring (P) and Marchigian Sardinian Alcohol-Preferring (msP) rats, without affecting food/water intake or locomotor activity.
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文献和实验个CD序号。 表6-1 抗人白细胞分化抗原McAb分组 分组 CD编号 T细胞 CD1~CD8,CD27,CD28,CD60,CD98~CDw101 B细胞 CD10,CD19~CD24,CD37,CD39,CD40,CD72~CD86 活化细胞 CD25,CDw26,CD30,CD69~CD71,CD95~CD97 髓样细胞 CD9,CD11b~CD17,CD31~CD36,CD64~CD68,CD87~CD93,CD115 NK/非谱系细胞 CD11a,CD18,CD29,CD
97 髓样细胞 CD9,CD11b~CD17,CD31~CD36,CD64~CD68,CD87~CD93,CD115 NK/非谱系细胞 CD11a,CD18,CD29,CD38,CD43,CE45~CD48,CD52~CD59,CD94 血小板 CD41,CD42,CD63,CD107 内皮
in playing a functional role in developmental stem cell biology (see reference 42 for a review). Sca-1 : Sca-1 (stem cell antigen 1, Ly-6A/E), an 18 kDa phosphatidylinositol-anchored protein, is a member of the Ly-6 antigen family.43 Sca
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